SCHEMBL5859258

SCHEMBL5859258

COC1=C(OC)C(=O)C(c2cc(C)c(-c3ccncc3)c(C(=O)N3CCOCC3)c2)=C(C)C1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
KDM4E B2RXH2 3/20 0.40
LMNA P02545 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPK1 P28482 1/20 0.39
LRRK2 Q5S007 1/20 0.39
CYP46A1 Q9Y6A2 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PLAUR Q03405 1/20 0.38
PKM P14618 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TSHR P16473 1/20 0.38
TP53 P04637 1/20 0.38
RAB9A P51151 2/20 0.37
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
TYK2 P29597 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5862104 0.91 PLAUR (0.44) ALDH1A1KDM4ELMNAMEN1KMT2A
SCHEMBL5862246 0.90 CYP2C9 (0.41) ALDH1A1KDM4EMEN1KMT2ACYP46A1
SCHEMBL5859257 0.90 HTT (0.45) ALDH1A1KDM4EMEN1KMT2AMAPK1
SCHEMBL5859916 0.90 RAB9A (0.49) ALDH1A1KDM4EMEN1KMT2AL3MBTL1
SCHEMBL5859907 0.86 RAB9A (0.49) ALDH1A1KDM4EMEN1KMT2AMAPK1
SCHEMBL5859860 0.82 IKBKB (0.37) KDM4ECYP46A1
SCHEMBL5859929 0.81 TDP1 (0.41) TSHRRAB9AHTTSMN1; SMN2NPC1
SCHEMBL5859235 0.80 CYP2C9 (0.45) ALDH1A1MEN1KMT2AHPGDTP53
SCHEMBL5859859 0.80 TDP1 (0.46) ALDH1A1KDM4ELMNAGAAHPGD
SCHEMBL7063575 0.79 JAK2 (0.40) KDM4ELMNAJAK2JAK1TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7122543-B2 Substituted benzoic acid derivatives having NF-κB inhibiting action DAIICHI SUNTORY PHARMA CO., LTD. (JP) 2006-10-17 US disclosed
EP-1437339-A1 SUBSTITUTED BENZOIC ACID DERIVATIVES EXHIBITING NF-KAPPA B INHIBITING ACTIVITY Daiichi Suntory Pharma Co., Ltd. (JP) 2004-07-14 EP disclosed