SCHEMBL5860481

SCHEMBL5860481

[CH2]c1cc(Cl)c(C(F)(F)F)cc1[N+](=O)[O-]

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.47
TSHR P16473 4/20 0.47
ALDH1A1 P00352 4/20 0.47
TDP1 Q9NUW8 3/20 0.47
ALOX15 P16050 2/20 0.47
HPGD P15428 1/20 0.47
HIF1A Q16665 1/20 0.47
TXNRD1 Q16881 1/20 0.47
TXNRD3 Q86VQ6 1/20 0.47
TXNRD2 Q9NNW7 1/20 0.47
MAPK1 P28482 3/20 0.38
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37
CCR2 P41597 1/20 0.36
SIRT6 Q8N6T7 1/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP2D6 P10635 1/20 0.35
GPR35 Q9HC97 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL602444 0.84 TSHR (0.52) CYP3A4TSHRALDH1A1TDP1ALOX15
SCHEMBL29672221 0.84 TSHR (0.52) CYP3A4TSHRALDH1A1TDP1ALOX15
SCHEMBL1770903 0.81 ALDH1A1 (0.49) CYP3A4TSHRALDH1A1TDP1ALOX15
SCHEMBL29435964 0.81 ALDH1A1 (0.49) CYP3A4TSHRALDH1A1TDP1ALOX15
SCHEMBL1770886 0.79 TSHR (0.47) CYP3A4TSHRALDH1A1TDP1ALOX15
SCHEMBL29672268 0.79 ALDH1A1 (0.47) CYP3A4TSHRALDH1A1TDP1ALOX15
SCHEMBL313585 0.79 ALDH1A1 (0.49) CYP3A4TSHRALDH1A1TDP1ALOX15
SCHEMBL29937444 0.79 TSHR (0.47) CYP3A4TSHRALDH1A1TDP1ALOX15
SCHEMBL1024954 0.79 ALDH1A1 (0.47) CYP3A4TSHRALDH1A1TDP1ALOX15
SCHEMBL10400092 0.79 TSHR (0.47) CYP3A4TSHRALDH1A1TDP1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7012146-B2 Ion channel modulating agents POSEIDON PHARMACEUTICALS A/S (DK) 2006-03-14 US claimed
US-20020169203-A1 Ion channel modulating agents NEUROSEARCH A/S (DK) 2002-11-14 US claimed
EP-1140784-A2 ION CHANNEL MODULATING AGENTS NEUROSEARCH A/S (DK) 2001-10-10 EP claimed
WO-2000037422-A2 ION CHANNEL MODULATING AGENTS NEUROSEARCH A/S (DK) 2000-06-29 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020169203-A1 Ion channel modulating agents KCNN3, KCNN1, KCNN2 CYP3A4 4157/4885TSHR 4434/4885ALDH1A1 4482/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.