SCHEMBL586094

SCHEMBL586094

N#Cc1c[nH]c2cccnc12

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 3/20 0.54
IMPDH2 P12268 1/20 0.52
IMPDH1 P20839 1/20 0.52
KCNMA1 Q12791 10/20 0.47
PSMD14 O00487 1/20 0.44
GRM4 Q14833 3/20 0.41
CCNT1 O60563 1/20 0.40
CDK9 P50750 1/20 0.40
HASPIN Q8TF76 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30186073 1.00 LRRK2 (0.54) LRRK2IMPDH2IMPDH1KCNMA1PSMD14
SCHEMBL29112310 0.76 LRRK2 (0.57) LRRK2IMPDH2IMPDH1CDK9
SCHEMBL19606882 0.75 PSMD14 (0.39) LRRK2IMPDH2IMPDH1KCNMA1PSMD14
SCHEMBL3887037 0.74 CSNK2A1 (0.46) LRRK2KCNMA1PSMD14GRM4
SCHEMBL11167116 0.74 PSMD14 (0.41) LRRK2KCNMA1PSMD14GRM4
SCHEMBL30052607 0.73 IMPDH2 (0.42) LRRK2IMPDH2IMPDH1CCNT1CDK9
SCHEMBL31586447 0.73 IMPDH2 (0.42) LRRK2IMPDH2IMPDH1CCNT1CDK9
SCHEMBL19273386 0.73 KCNMA1 (0.41) LRRK2KCNMA1PSMD14GRM4
SCHEMBL31588050 0.72 PARP1 (0.50) LRRK2IMPDH2IMPDH1
SCHEMBL10254 0.72 PARP1 (0.50) LRRK2IMPDH2IMPDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417133-A1 COMPOUNDS AND METHODS FOR ANTIVIRAL TREATMENT PTC Therapeutics, Inc. (US) 2012-02-15 EP disclosed
WO-2010117935-A1 COMPOUNDS AND METHODS FOR ANTIVIRAL TREATMENT SCHERING CORPORATION (US) 2010-10-14 WO disclosed