SCHEMBL5862792

SCHEMBL5862792

COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1

nearest known ligand 0.72

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.72
CCR5 P51681 10/20 0.72
SIGMAR1 Q99720 2/20 0.65
CHRM2 P08172 2/20 0.62
CHRM3 P20309 2/20 0.62
GPR119 Q8TDV5 2/20 0.56
MCHR1 Q99705 1/20 0.56
FAAH O00519 1/20 0.55
ACHE P22303 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6703964 0.86 KCNH2 (0.79) KCNH2CCR5SIGMAR1CHRM2CHRM3
SCHEMBL19658476 0.83 CHRM2 (0.57) KCNH2CCR5SIGMAR1CHRM2CHRM3
SCHEMBL4220408 0.83 OPRM1 (0.63) KCNH2CCR5SIGMAR1CHRM2CHRM3
SCHEMBL2405257 0.83 CCR5 (0.62) CCR5SIGMAR1
Hydrochloric Acid SCHEMBL4920052 0.82 OPRM1 (0.62) KCNH2CCR5SIGMAR1CHRM2CHRM3
Oxalic Acid SCHEMBL4217435 0.81 OPRM1 (0.61) KCNH2CCR5SIGMAR1CHRM2CHRM3
SCHEMBL339984 0.81 SIGMAR1 (0.58) KCNH2CCR5SIGMAR1CHRM2CHRM3
SCHEMBL339985 0.81 SIGMAR1 (0.58) KCNH2CCR5SIGMAR1CHRM2CHRM3
SCHEMBL13478882 0.80 KCNH2 (0.67) KCNH2CCR5SIGMAR1CHRM2CHRM3
SCHEMBL5116528 0.80 KCNH2 (0.67) KCNH2CCR5SIGMAR1CHRM2CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7041667-B1 CCR5 modulators PFIZER, INC. (US) 2006-05-09 US disclosed