SCHEMBL5864840

SCHEMBL5864840

COc1cccc2c1CCC(c1cc(N)ccn1)=C2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ASIC3 Q9UHC3 3/20 0.38
KDM4C Q9H3R0 1/20 0.36
OPRD1 P41143 1/20 0.36
KCNH2 Q12809 1/20 0.36
ADRA2A P08913 1/20 0.35
ADRA1A P35348 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
RAB9A P51151 1/20 0.35
DYRK1A Q13627 2/20 0.34
HTR1A P08908 1/20 0.34
HTR7 P34969 1/20 0.34
HTR2B P41595 1/20 0.34
HTR5A P47898 1/20 0.34
NFATC1 O95644 1/20 0.34
GSK3B P49841 1/20 0.34
CYP19A1 P11511 1/20 0.34
GRM5 P41594 2/20 0.34
GRM1 Q13255 2/20 0.34
APLNR P35414 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL5864807 0.90 KDM4C (0.39) ASIC3KDM4COPRD1KCNH2KDM4E
Fumaric Acid SCHEMBL5864817 0.90 KDM4C (0.39) ASIC3KDM4COPRD1KCNH2KDM4E
SCHEMBL5865110 0.75 ASIC3 (0.47) ASIC3OPRD1ADRA1AKDM4EALDH1A1
SCHEMBL5864811 0.75 KDM1A (0.34) ALDH1A1RAB9ACYP19A1
SCHEMBL5865162 0.74 CYP11B2 (0.54) ASIC3OPRD1KCNH2KDM4EALDH1A1
Hydrochloric Acid SCHEMBL5865331 0.74 ASIC3 (0.46) ASIC3OPRD1ADRA1AKDM4EALDH1A1
SCHEMBL5865078 0.74 ASIC3 (0.36) ASIC3KDM4E
SCHEMBL5865045 0.73 ASIC3 (0.38) ASIC3ALDH1A1
SCHEMBL22558013 0.71 PTGS2 (0.45) ALDH1A1RAB9ACYP19A1PTGS2
SCHEMBL28452211 0.70 HSP90AA1 (0.53) ASIC3KDM4CKDM4EALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7034044-B2 Conjugated aromatic compounds with a pyridine substituent HOFFMANN-LA ROCHE INC. (US) 2006-04-25 US disclosed
US-20060058354-A1 Conjugated aromatic compounds with a pyridine substituent ALANINE ALEXANDER 2006-03-16 US disclosed
US-6951875-B2 Conjugated aromatic compounds with a pyridine substituent HOFFMANN-LA ROCHE INC. (US) 2005-10-04 US disclosed
US-20040068118-A1 Conjugated aromatic compounds with a pyridine substituent ALANINE ALEXANDER (FR) 2004-04-08 US disclosed
US-20030144525-A1 Conjugated aromatic compounds with a pyridine substituent HOFFMANN-LA ROCHE INC. 2003-07-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040068118-A1 Conjugated aromatic compounds with a pyridine substituent GRIN2B, GRIN1, GRIN2C ASIC3 463/4885KDM4C 994/4885OPRD1 163/4885
US-20030144525-A1 Conjugated aromatic compounds with a pyridine substituent GRIN2B, GRIN1, GRIN2C ASIC3 463/4885KDM4C 994/4885OPRD1 163/4885
US-20060058354-A1 Conjugated aromatic compounds with a pyridine substituent GRIN2B, GRIN3A, GRIN2C ASIC3 502/4885KDM4C 777/4885OPRD1 218/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.