SCHEMBL5869169

SCHEMBL5869169

Sc1cccc2ccsc12

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.50
HDAC4 P56524 1/20 0.40
PSMD14 O00487 2/20 0.35
COPS5 Q92905 2/20 0.35
DAO P14920 1/20 0.35
PIM1 P11309 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
HDAC1 Q13547 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
CYP19A1 P11511 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3799554 0.71 CYP2A6 (0.50) CYP2A6HDAC4DAOPIM1SLC6A2
SCHEMBL276295 0.71 CYP2A6 (0.55) CYP2A6HDAC4DAOPIM1SLC6A2
SCHEMBL1866237 0.71 CYP2A6 (0.50) CYP2A6HDAC4DAOPIM1SLC6A2
SCHEMBL14022908 0.71 CYP2A6 (0.50) CYP2A6HDAC4DAOPIM1SLC6A2
SCHEMBL389275 0.71 CYP2A6 (0.50) CYP2A6HDAC4DAOPIM1SLC6A2
SCHEMBL156699 0.71 CYP2A6 (0.50) CYP2A6HDAC4DAOPIM1SLC6A2
SCHEMBL911242 0.71 CYP2A6 (0.50) CYP2A6HDAC4DAOPIM1SLC6A2
SCHEMBL594318 0.71 CYP2A6 (0.50) CYP2A6HDAC4DAOPIM1SLC6A2
SCHEMBL2011067 0.71 CYP2A6 (0.50) CYP2A6HDAC4DAOPIM1SLC6A2
SCHEMBL288299 0.71 CYP2A6 (0.50) CYP2A6HDAC4DAOPIM1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111057074-B Inhibitors of influenza virus replication and uses thereof 广东东阳光药业有限公司 2022-04-29 CN disclosed
CN-111057074-A Inhibitors of influenza virus replication and uses thereof 广东东阳光药业有限公司 2020-04-24 CN disclosed
US-7037932-B2 Heteroaryloxy 3-substituted propanamines as serotonin and norepinephrine reuptake inhibitors ELI LILLY AND COMPANY (US) 2006-05-02 US disclosed
EP-1397129-B1 HETEROARYLOXY 3-SUBSTITUTED PROPANAMINES S SEROTONIN AND NOREPINEPHRINE REUPTAKE INHIBITORS LILLY CO ELI (US) 2005-11-16 EP disclosed
US-20040176435-A1 Heteroaryloxy 3-substituted propanamines s serotonin and norepinephrine reuptake inhibitors ELI LILLY AND COMPANY 2004-09-09 US disclosed
EP-1397129-A1 HETEROARYLOXY 3-SUBSTITUTED PROPANAMINES S SEROTONIN AND NOREPINEPHRINE REUPTAKE INHIBITORS ELI LILLY AND COMPANY (US) 2004-03-17 EP disclosed
WO-2002094262-A1 HETEROARYLOXY 3-SUBSTITUTED PROPANAMINES S SEROTONIN AND NOREPINEPHRINE REUPTAKE INHIBITORS ELI LILLY AND COMPANY (US) 2002-11-28 WO disclosed
US-5730860-A USING ABSORBENT; COUNTERCURRENT FLOW THE PRITCHARD CORPORATION (US) 1998-03-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040176435-A1 Heteroaryloxy 3-substituted propanamines s serotonin and norepinephrine reuptake inhibitors ADRA2C, ADRB1, TPH1 CYP2A6 178/4885HDAC4 1135/4885PSMD14 4252/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.