SCHEMBL5869563

SCHEMBL5869563

COC(=O)C(Cc1ccc([N+](=O)[O-])cn1)NC(=O)OC(C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSTP1 P09211 1/20 0.50
GSTM2 P28161 1/20 0.50
CYP2C19 P33261 2/20 0.47
PPARG P37231 1/20 0.46
PPARA Q07869 1/20 0.46
KLK5 Q9Y337 1/20 0.41
ITGA4 P13612 1/20 0.40
ITGB7 P26010 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.39
NPC1 O15118 3/20 0.39
MAPT P10636 3/20 0.39
RAB9A P51151 3/20 0.39
ALDH1A1 P00352 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
GAA P10253 2/20 0.39
CYP1A2 P05177 1/20 0.38
LMNA P02545 1/20 0.38
KDM4E B2RXH2 1/20 0.38
HDAC6 Q9UBN7 4/20 0.37
HDAC1 Q13547 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5147742 0.92 PPARG (0.45) GSTP1GSTM2CYP2C19PPARGPPARA
SCHEMBL2983423 0.90 PPARA (0.54) GSTP1GSTM2CYP2C19PPARGPPARA
SCHEMBL27589045 0.90 PPARA (0.54) GSTP1GSTM2CYP2C19PPARGPPARA
SCHEMBL2983425 0.90 PPARA (0.54) GSTP1GSTM2CYP2C19PPARGPPARA
SCHEMBL3319460 0.83 PPARG (0.58) GSTP1GSTM2PPARGPPARAKLK5
SCHEMBL19212613 0.83 PPARG (0.58) GSTP1GSTM2PPARGPPARAKLK5
SCHEMBL2728823 0.83 PPARG (0.58) GSTP1GSTM2PPARGPPARAKLK5
SCHEMBL4074909 0.83 CTSS (0.46) GSTP1GSTM2PPARAKLK5HDAC6
SCHEMBL16645014 0.83 KLK5 (0.45) GSTP1GSTM2PPARGPPARAKLK5
SCHEMBL8232460 0.83 KLK5 (0.45) GSTP1GSTM2PPARGPPARAKLK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7045532-B2 ACE-2 modulating compounds and methods of use thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2006-05-16 US disclosed
US-20040082496-A1 ACE-2 modulating compounds and methods of use thereof MILLENNIUM PHARMACEUTICALS, INC. 2004-04-29 US disclosed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040082496-A1 ACE-2 modulating compounds and methods of use thereof ACE, ACE2, AGTR2 GSTP1 399/4885GSTM2 307/4885CYP2C19 1489/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.