SCHEMBL5871916

SCHEMBL5871916

COC(=O)C(=Cc1[c]ccc(C(F)(F)F)c1)C(=O)OC

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.38
GPR35 Q9HC97 1/20 0.38
GAA P10253 2/20 0.37
MAPT P10636 2/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5872067 0.79 MAPT (0.40) MAPTLMNAHPGD
SCHEMBL5871857 0.79 MAPT (0.40) MAPTLMNAHPGD
SCHEMBL5871437 0.79 MAPT (0.40) MAPTALDH1A1LMNAHPGD
SCHEMBL5871896 0.78 MAPT (0.42) MAPTALDH1A1HPGD
SCHEMBL23668754 0.78 MAPT (0.39) GAAMAPTLMNAHPGD
SCHEMBL5872103 0.74 MAPT (0.42) GAAMAPTLMNAHPGD
SCHEMBL5871874 0.72 MAPT (0.46) MAPTLMNAHPGD
SCHEMBL27844712 0.71 CES2 (0.33) MAPTALDH1A1HPGD
SCHEMBL5551833 0.71 CFTR (0.50) CFTRGAAMAPTALDH1A1LMNA
SCHEMBL5871435 0.70 PTPRB (0.38) CFTRGAAMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7071187-B2 Naphthyridine derivatives OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 2006-07-04 US disclosed
US-20040214853-A1 Naphthyridine derivatives OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 2004-10-28 US disclosed
EP-1426374-A1 NAPHTHYRIDINE DERIVATIVE OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 2004-06-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040214853-A1 Naphthyridine derivatives MT-ND1, OPRD1, NR0B1 CFTR 3918/4885GPR35 1694/4885GAA 1753/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.