SCHEMBL5873340

SCHEMBL5873340

COc1cc2c(cc1OC)N(Cc1ccccc1)CCN=C2c1cccc(C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK10 P53779 5/20 0.43
THRB P10828 1/20 0.40
PDE4B Q07343 1/20 0.39
HTR1D P28221 1/20 0.39
HTR1B P28222 1/20 0.39
GPR55 Q9Y2T6 1/20 0.39
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
CXCR2 P25025 1/20 0.39
PTAFR P25105 1/20 0.38
GRM5 P41594 1/20 0.38
GRM1 Q13255 1/20 0.38
NPC1 O15118 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38
NR1I2 O75469 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
HTR2C P28335 1/20 0.38
ADRA1A P35348 1/20 0.38
PTGS2 P35354 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4710191 0.81 NPSR1 (0.58) GPR55GRM5GRM1NR1I2ADORA3
SCHEMBL4709468 0.73 PDE2A (0.57) GRM5GRM1OPRK1
SCHEMBL4709481 0.73 GRM5 (0.47) PDE4BGPR55GRM5GRM1GRIN1
SCHEMBL4707946 0.71 GRM5 (0.46) PDE4BGPR55GRM5GRM1GRIN1
SCHEMBL4709544 0.70 NPSR1 (0.47) THRBGPR55BCHEACHEGRM5
SCHEMBL5368722 0.69 SIGMAR1 (0.47) MAPK10GPR55NR1I2ADORA3HTR2C
SCHEMBL5492932 0.67 TP53 (0.60) GPR55
SCHEMBL4709565 0.67 NPSR1 (0.56) GPR55GRM5GRM1NR1I2ADORA3
SCHEMBL11679315 0.67 OPRK1 (0.67) PTAFRNR1I2ADORA3HTR2CADRA1A
SCHEMBL4710060 0.66 TUBB4A (0.50) PDE4BGRM5GRM1OPRK1PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006509832-A 2006-03-23 JP claimed
EP-1556055-A2 USE OF CYCLIC NUCLEOTIDE PHOSPHODIESTERASE INHIBITORS HAVING A BENZODIAZEPINE STRUCTURE IN THERAPY NEURO3D (FR) 2005-07-27 EP claimed
WO-2004041258-A2 CYCLIC NUCLEOTIDE PHOSPHODIESTERASE INHIBITORS, PREPARATION AND USES NEURO3D (FR) 2004-05-21 WO claimed