SCHEMBL587434

SCHEMBL587434

COC(=O)C1CCN(C(=O)OC)C(Cc2cc(C(C)(C)C)cc(C(C)(C)C)c2)C1.COC(=O)N1CCC(C(=O)O)CC1Cc1cc(C(C)(C)C)cc(C(C)(C)C)c1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.39
ALDH1A1 P00352 5/20 0.37
MAPT P10636 3/20 0.37
NPSR1 Q6W5P4 2/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
TACR1 P25103 7/20 0.36
CETP P11597 2/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
CYP3A4 P08684 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HTT P42858 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
NEK2 P51955 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL587545 0.96 OPRK1 (0.42) OPRK1ALDH1A1MAPTNPSR1HPGD
SCHEMBL581245 0.96 TACR1 (0.38) OPRK1ALDH1A1MAPTNPSR1HPGD
SCHEMBL581020 0.85 OPRK1 (0.35) OPRK1ALDH1A1MAPTNPSR1HPGD
SCHEMBL581238 0.85 NPC1 (0.41) ALDH1A1HSD17B10TACR1NPC1RAB9A
SCHEMBL3081551 0.84 TACR1 (0.39) ALDH1A1NPSR1HPGDHSD17B10TACR1
SCHEMBL587423 0.83 TACR1 (0.45) ALDH1A1MAPTNPSR1HPGDHSD17B10
SCHEMBL587559 0.82 TACR1 (0.43) OPRK1ALDH1A1MAPTNPSR1HPGD
SCHEMBL3087575 0.81 MEN1 (0.36) ALDH1A1MAPTTACR1CETPNPC1
SCHEMBL581268 0.81 MEN1 (0.36) ALDH1A1MAPTTACR1CETPNPC1
SCHEMBL581269 0.81 MEN1 (0.36) ALDH1A1MAPTTACR1CETPNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed