SCHEMBL5876853

SCHEMBL5876853

COc1cc(-c2nc3ccc(Cl)cc3c(=O)n2CC2CCCC(CN)C2)cc(OC)c1OC

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 2/20 0.44
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CYP2D6 P10635 3/20 0.43
HTR2C P28335 1/20 0.43
GHSR Q92847 2/20 0.42
CYP3A4 P08684 1/20 0.42
KCNH2 Q12809 1/20 0.42
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ALOX5 P09917 1/20 0.39
AVPR1A P37288 1/20 0.39
EGFR P00533 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5877840 0.93 EGFR (0.45) ABCC1LMNASMN1; SMN2CYP2D6HTR2C
SCHEMBL5877641 0.91 ABCC1 (0.46) ABCC1CYP2D6HTR2CGHSRCYP3A4
SCHEMBL5877323 0.91 SMN1; SMN2 (0.45) ABCC1LMNASMN1; SMN2CYP2D6HTR2C
SCHEMBL5877465 0.90 LMNA (0.44) ABCC1LMNASMN1; SMN2CYP2D6GHSR
SCHEMBL5878058 0.88 SMN1; SMN2 (0.58) ABCC1LMNASMN1; SMN2CYP2D6MEN1
SCHEMBL5877561 0.88 CYP2D6 (0.46) ABCC1CYP2D6HTR2CGHSRCYP3A4
SCHEMBL5877425 0.86 CYP2D6 (0.43) ABCC1CYP2D6HTR2CGHSRCYP3A4
SCHEMBL5877998 0.85 MEN1 (0.53) ABCC1LMNACYP2D6HTR2CGHSR
SCHEMBL5877392 0.85 CYP2D6 (0.46) ABCC1CYP2D6HTR2CGHSRCYP3A4
SCHEMBL5878217 0.85 POLB (0.46) CYP2D6HTR2CGHSRCYP3A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060706-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed
EP-1216233-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023364-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed