SCHEMBL5877323

SCHEMBL5877323

COc1cc(-c2nc3ccc(C)cc3c(=O)n2CC2CCCC(CN)C2)cc(OC)c1OC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.45
LMNA P02545 1/20 0.45
ABCC1 P33527 2/20 0.40
MAP3K11 Q16584 1/20 0.39
PDE5A O76074 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
PNP P00491 1/20 0.38
CYP2D6 P10635 2/20 0.37
GHSR Q92847 2/20 0.37
HTR2C P28335 1/20 0.37
POLB P06746 1/20 0.37
KDM4E B2RXH2 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
CYP3A4 P08684 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5877465 0.92 LMNA (0.44) SMN1; SMN2LMNAABCC1MAP3K11CYP2D6
SCHEMBL5876853 0.91 ABCC1 (0.44) SMN1; SMN2LMNAABCC1CYP2D6GHSR
SCHEMBL5878313 0.91 PDE4B (0.43) SMN1; SMN2LMNAABCC1MAP3K11PDE4B
SCHEMBL5878058 0.90 SMN1; SMN2 (0.58) SMN1; SMN2LMNAABCC1CYP2D6POLB
SCHEMBL5877963 0.87 ALDH1A1 (0.47) SMN1; SMN2LMNAABCC1GHSRPOLB
SCHEMBL5876953 0.86 ABCC1 (0.50) SMN1; SMN2ABCC1CYP2D6GHSRHTR2C
SCHEMBL5877840 0.86 EGFR (0.45) SMN1; SMN2LMNAABCC1MAP3K11PDE5A
SCHEMBL5877626 0.86 ABCC1 (0.52) SMN1; SMN2ABCC1CYP2D6GHSRHTR2C
SCHEMBL5876985 0.85 CRHR1 (0.44) SMN1; SMN2LMNAABCC1CYP2D6GHSR
SCHEMBL5877811 0.85 ABCC1 (0.46) ABCC1CYP2D6GHSRHTR2CCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060706-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed