SCHEMBL5877425

SCHEMBL5877425

COc1ccc(-c2ccc(-c3nc4ccc(Cl)cc4c(=O)n3CC3CCCC(CN)C3)cc2)c(OC)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.43
HTR2C P28335 1/20 0.43
GHSR Q92847 3/20 0.43
KCNH2 Q12809 2/20 0.43
ABCC1 P33527 2/20 0.43
CYP3A4 P08684 1/20 0.43
CRHR1 P34998 1/20 0.42
F11 P03951 1/20 0.42
POLB P06746 2/20 0.42
RXFP1 Q9HBX9 1/20 0.42
ADRA1A P35348 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2B Q13224 1/20 0.41
ALOX5 P09917 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
AKR1B10 O60218 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5877807 0.94 F11 (0.47) CYP2D6HTR2CGHSRKCNH2ABCC1
SCHEMBL5877717 0.94 EGFR (0.44) CYP2D6HTR2CGHSRKCNH2ABCC1
SCHEMBL5877561 0.93 CYP2D6 (0.46) CYP2D6HTR2CGHSRKCNH2ABCC1
SCHEMBL5876985 0.92 CRHR1 (0.44) CYP2D6HTR2CGHSRKCNH2ABCC1
SCHEMBL5877906 0.89 ABCC1 (0.52) ABCC1CRHR1POLBRXFP1MEN1
SCHEMBL5877446 0.89 CRHR1 (0.41) CYP2D6HTR2CGHSRKCNH2CYP3A4
SCHEMBL5877392 0.88 CYP2D6 (0.46) CYP2D6HTR2CGHSRKCNH2ABCC1
SCHEMBL5877641 0.88 ABCC1 (0.46) CYP2D6HTR2CGHSRKCNH2ABCC1
SCHEMBL5876981 0.87 F11 (0.52) CYP2D6GHSRKCNH2ABCC1F11
SCHEMBL5878217 0.87 POLB (0.46) CYP2D6HTR2CGHSRKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060706-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed
EP-1216233-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023364-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed