SCHEMBL5877135

SCHEMBL5877135

CC(c1ccccc1)c1nc2ccccc2c(=O)n1CC1CCCC(CN)C1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 1/20 0.47
ALDH1A1 P00352 6/20 0.46
NPSR1 Q6W5P4 4/20 0.46
PLA2G1B P04054 1/20 0.46
ATG4B Q9Y4P1 1/20 0.46
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
LMNA P02545 2/20 0.41
HIF1A Q16665 2/20 0.41
HTT P42858 1/20 0.41
RECQL P46063 1/20 0.39
CYP2D6 P10635 3/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CACNA2D1 P54289 3/20 0.38
PDE7A Q13946 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5878279 0.90 CYP2D6 (0.45) ABCC1ALDH1A1NPSR1PLA2G1BATG4B
SCHEMBL5877929 0.89 CYP2D6 (0.42) ABCC1ALDH1A1NPSR1PLA2G1BATG4B
SCHEMBL5877630 0.88 CYP2D6 (0.49) ABCC1CYP2D6
SCHEMBL5877473 0.87 CYP2D6 (0.46) ALDH1A1NPSR1PLA2G1BATG4BLMNA
SCHEMBL5877050 0.81 ABCC1 (0.62) ABCC1ALDH1A1NPSR1PLA2G1BATG4B
SCHEMBL5877489 0.80 ABCC1 (0.53) ABCC1ALDH1A1NPSR1PLA2G1BATG4B
SCHEMBL5878320 0.80 ABCC1 (0.62) ABCC1ALDH1A1NPSR1TDP1L3MBTL1
SCHEMBL5877881 0.78 ABCC1 (0.53) ABCC1ALDH1A1NPSR1PLA2G1BATG4B
SCHEMBL5877284 0.78 ATM (0.58) ABCC1ALDH1A1NPSR1PLA2G1BATG4B
SCHEMBL5878390 0.77 ABCC1 (0.59) ABCC1ALDH1A1NPSR1PLA2G1BATG4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060706-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed
EP-1216233-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023364-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed