SCHEMBL5877929

SCHEMBL5877929

Cc1ccc2nc(C(C)c3ccccc3)n(CC3CCCC(CN)C3)c(=O)c2c1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 7/20 0.42
GHSR Q92847 5/20 0.41
KCNH2 Q12809 2/20 0.41
CYP3A4 P08684 1/20 0.41
ABCC1 P33527 1/20 0.39
ALDH1A1 P00352 1/20 0.39
PLA2G1B P04054 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ATG4B Q9Y4P1 1/20 0.39
HTR2C P28335 1/20 0.38
DHFR P00374 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ALOX5AP P20292 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5877630 0.90 CYP2D6 (0.49) CYP2D6GHSRKCNH2CYP3A4ABCC1
SCHEMBL5877135 0.89 ABCC1 (0.47) CYP2D6ABCC1ALDH1A1PLA2G1BNPSR1
SCHEMBL5877473 0.88 CYP2D6 (0.46) CYP2D6GHSRKCNH2CYP3A4ALDH1A1
SCHEMBL5877626 0.85 ABCC1 (0.52) CYP2D6GHSRKCNH2CYP3A4ABCC1
SCHEMBL5878279 0.85 CYP2D6 (0.45) CYP2D6GHSRKCNH2CYP3A4ABCC1
SCHEMBL5877732 0.83 ABCC1 (0.52) CYP2D6GHSRKCNH2CYP3A4ABCC1
SCHEMBL5877867 0.83 GHSR (0.54) CYP2D6GHSRKCNH2CYP3A4ABCC1
SCHEMBL5877811 0.82 ABCC1 (0.46) CYP2D6GHSRKCNH2CYP3A4ABCC1
SCHEMBL5876953 0.82 ABCC1 (0.50) CYP2D6GHSRKCNH2CYP3A4ABCC1
SCHEMBL5877870 0.81 ABCC1 (0.48) CYP2D6GHSRKCNH2CYP3A4ABCC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060706-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed