SCHEMBL5877473

SCHEMBL5877473

COc1ccc2nc(C(C)c3ccccc3)n(CC3CCCC(CN)C3)c(=O)c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 5/20 0.46
LMNA P02545 1/20 0.45
RECQL P46063 1/20 0.45
DPP4 P27487 2/20 0.43
CYP3A4 P08684 2/20 0.43
ADORA3 P0DMS8 3/20 0.42
GHSR Q92847 5/20 0.41
TUBB4A P04350 1/20 0.41
TUBB P07437 1/20 0.41
TUBA3C P0DPH7 1/20 0.41
TUBA1B P68363 1/20 0.41
TUBA4A P68366 1/20 0.41
TUBB4B P68371 1/20 0.41
TUBB3 Q13509 1/20 0.41
TUBB2A Q13885 1/20 0.41
TUBB8 Q3ZCM7 1/20 0.41
TUBA3E Q6PEY2 1/20 0.41
TUBA1A Q71U36 1/20 0.41
TUBA1C Q9BQE3 1/20 0.41
TUBB6 Q9BUF5 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5877929 0.88 CYP2D6 (0.42) CYP2D6CYP3A4GHSRKCNH2ALOX5AP
SCHEMBL5877630 0.87 CYP2D6 (0.49) CYP2D6DPP4CYP3A4GHSRTUBB4A
SCHEMBL5877135 0.87 ABCC1 (0.47) CYP2D6LMNARECQLALDH1A1PLA2G1B
SCHEMBL5877978 0.85 AVPR1B (0.49) CYP2D6GHSRKCNH2AVPR1BHRH3
SCHEMBL5877069 0.84 F11 (0.49) CYP2D6CYP3A4GHSRKCNH2AVPR1B
SCHEMBL5877494 0.83 GHSR (0.60) CYP2D6DPP4CYP3A4ADORA3GHSR
SCHEMBL5878279 0.83 CYP2D6 (0.45) CYP2D6DPP4CYP3A4GHSRKCNH2
SCHEMBL5876981 0.82 F11 (0.52) CYP2D6LMNAGHSRKCNH2AVPR1B
SCHEMBL5877542 0.82 F11 (0.46) CYP2D6DPP4CYP3A4GHSRKCNH2
SCHEMBL5877712 0.82 AVPR1B (0.51) GHSRAVPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060706-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed
EP-1216233-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023364-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed