SCHEMBL5877529

SCHEMBL5877529

Cc1ccc(S(=O)(=O)n2nc(NC3CC3)c3c2CC(c2cccnc2)(c2cccnc2)C=C3)cc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
ALDH1A1 P00352 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 1/20 0.35
CCR6 P51684 2/20 0.34
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
PKM P14618 1/20 0.33
GFER P55789 1/20 0.33
POLB P06746 1/20 0.32
GPR6 P46095 1/20 0.32
TSHR P16473 1/20 0.32
EGFR P00533 1/20 0.31
PTGS2 P35354 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5877112 0.97 ALDH1A1 (0.37) CYP3A4CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL5876940 0.97 CYP3A4 (0.35) CYP3A4CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL5877418 0.94 ALDH1A1 (0.36) CYP3A4CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL5876012 0.90 NR1H2 (0.36) CYP2C19ALDH1A1CCR6GPR6
SCHEMBL5876220 0.90 NR1H2 (0.34) CYP2C19ALDH1A1LMNACCR6GPR6
SCHEMBL5876928 0.89 CCR6 (0.34) ALDH1A1LMNACCR6POLBGPR6
SCHEMBL5876198 0.86 USP2 (0.37) CYP2C19ALDH1A1LMNACCR6TSHR
SCHEMBL5876674 0.86 USP2 (0.35) CYP2C19ALDH1A1CCR6TSHR
SCHEMBL5876433 0.86 POLB (0.36) CYP3A4CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL5877652 0.86 ACHE (0.34) CYP3A4ALDH1A1LMNACCR6POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7119115-B2 Indazole or indole derivatives, and use thereof in human medicine and more particularly in oncology AVENTIS PHARMA S.A. (FR) 2006-10-10 US disclosed
US-20040162276-A1 Indazole or indole derivatives, and use thereof in human medicine and more particularly in oncology AVENTIS PHARMA S.A. (FR) 2004-08-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040162276-A1 Indazole or indole derivatives, and use thereof in human medicine and more particularly in oncology IDO1, IDO2, INMT CYP3A4 26/4885CYP2D6 23/4885CYP2C9 44/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.