SCHEMBL5878

SCHEMBL5878

Fc1ccc(OBOc2ccc(F)cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 1/20 0.39
SOS1 Q07889 1/20 0.37
HSPB1 P04792 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
ACHE P22303 1/20 0.36
MAOB P27338 5/20 0.35
APP P05067 1/20 0.35
GAA P10253 1/20 0.34
IDO1 P14902 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
MAOA P21397 1/20 0.33
AGXT P21549 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
TDO2 P48775 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1758367 0.92 SOS1 (0.47) NFE2L2SOS1HSPB1GAAKDM4E
SCHEMBL3318479 0.90 LTA4H (0.40) NFE2L2MAOAMEN1KMT2A
SCHEMBL18670944 0.78 NFE2L2 (0.37) NFE2L2SOS1HSPB1CA1CA2
SCHEMBL121643 0.78 NFE2L2 (0.37) NFE2L2SOS1HSPB1CA1CA2
SCHEMBL6647494 0.76 SOS1 (0.39) NFE2L2SOS1CA1CA2CA7
SCHEMBL6867335 0.76 ALDH1A1 (0.48) SOS1HSPB1MAOBGAAMEN1
SCHEMBL5710196 0.76 NFE2L2 (0.35) NFE2L2SOS1HSPB1CA1CA2
SCHEMBL15234506 0.72 BCL2L1 (0.40) NFE2L2MAOBNPC1RAB9AMAOA
SCHEMBL17721283 0.72 SOS1 (0.44) SOS1HSPB1GAAKDM4EMEN1
SCHEMBL6289867 0.71 SOS1 (0.58) NFE2L2SOS1HSPB1GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2287 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240092822-A1 PURIFICATION METHODS FOR OLIGOMERIC COMPOUNDS IONIS PHARMACEUTICALS, INC. (US) 2024-03-21 US claimed
EP-4301766-A1 PURIFICATION METHODS FOR OLIGOMERIC COMPOUNDS Ionis Pharmaceuticals, Inc. (US) 2024-01-10 EP claimed
CN-115155640-B Molybdenum catalyst, catalytic composition and application thereof in preparation of amine compounds 海南华瑞医药有限公司 2023-09-05 CN claimed
US-11495769-B2 Inorganic light emitting diode and inorganic light emitting device including the same LG DISPLAY CO., LTD. (KR) 2022-11-08 US claimed
US-20210167321-A1 INORGANIC LIGHT EMITTING DIODE AND INORGANIC LIGHT EMITTING DEVICE INCLUDING THE SAME LG DISPLAY CO., LTD. (KR) 2021-06-03 US claimed
CN-111629746-A Charge switchable polymer depot for glucose triggered insulin delivery with ultra-fast response 北卡罗来纳州立大学 2020-09-04 CN claimed
EP-3134419-B1 NON-ENZYMATIC ELECTROCHEMICAL SENSOR FOR MEASURING ANALYTES TERUMO CORP (JP) 2019-03-13 EP claimed
US-20170219521-A1 NON-ENZYMATIC ELECTROCHEMICAL SENSOR FOR MEASURING ANALYTES TERUMO KABUSHIKI KAISHA (JP) 2017-08-03 US claimed
EP-3134419-A2 NON-ENZYMATIC ELECTROCHEMICAL SENSOR FOR MEASURING ANALYTES Glucovation, Inc. (US) 2017-03-01 EP claimed
WO-2015164578-A9 NON-ENZYMATIC ELECTROCHEMICAL SENSOR FOR MEASURING ANALYTES GLUCOVATION, INC. (US) 2016-02-18 WO claimed
WO-2015164578-A2 NON-ENZYMATIC ELECTROCHEMICAL SENSOR FOR MEASURING ANALYTES GLUCOVATION, INC. (US) 2015-10-29 WO claimed
US-8921299-B2 Detergents having acceptable color THE PROCTER & GAMBLE COMPANY (US) 2014-12-30 US claimed
EP-1064286-A1 SYNTHESIS OF ARYL BORONIC ACIDS BOULDER SCIENTIFIC COMPANY (US) 2001-01-03 EP claimed
WO-1999064428-A1 SYNTHESIS OF ARYL BORONIC ACIDS BOULDER SCIENTIFIC COMPANY (US) 1999-12-16 WO claimed
WO-1995005081-A1 BIOCIDAL COMPOSITIONS CONTAINING ORGANOBORON COMPOUNDS U.S. BORAX INC. (US) 1995-02-23 WO claimed
CN-116969925-B Heteroaryl-triazole compounds BAYER AG (DE) 2026-05-26 CN disclosed
CN-115835909-B Cannabinoid receptor type 2 (CB 2) modulators and uses thereof 泰昂治疗公司 2026-05-15 CN disclosed
EP-0544488-A2 Substituted phenyl phenol leukotriene antagonists ELI LILLY AND COMPANY (US) 1993-06-02 EP disclosed
EP-0413785-A1 LIQUID CRYSTALLINE MEDIA CONTAINING FLUORINATED OLIGOPHENYLS. MERCK PATENT GMBH (DE) 1991-02-27 EP disclosed
WO-1990009420-A1 LIQUID CRYSTALLINE MEDIA CONTAINING FLUORINATED OLIGOPHENYLS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1990-08-23 WO disclosed