SCHEMBL5878151

SCHEMBL5878151

COc1ccc2nc(-c3cccc4ccccc34)n(CC3CCCC(CN)C3)c(=O)c2c1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 9/20 0.50
CYP2D6 P10635 2/20 0.48
ABCC1 P33527 1/20 0.43
HTR2C P28335 1/20 0.43
KCNH2 Q12809 5/20 0.42
CYP3A4 P08684 2/20 0.42
ADORA3 P0DMS8 1/20 0.42
CYP1A1 P04798 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP1B1 Q16678 1/20 0.41
DPP4 P27487 1/20 0.41
GLA P06280 1/20 0.40
CRHR1 P34998 1/20 0.40
ADRA1A P35348 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
ACHE P22303 1/20 0.40
F11 P03951 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5877494 0.91 GHSR (0.60) GHSRCYP2D6ABCC1HTR2CKCNH2
SCHEMBL5878659 0.89 ABCC1 (0.46) GHSRCYP2D6ABCC1HTR2CKCNH2
SCHEMBL5877978 0.88 AVPR1B (0.49) GHSRCYP2D6ABCC1KCNH2ADRA1A
SCHEMBL5877881 0.87 ABCC1 (0.53) GHSRCYP2D6ABCC1HTR2CKCNH2
SCHEMBL5877542 0.87 F11 (0.46) GHSRCYP2D6ABCC1HTR2CKCNH2
SCHEMBL5877712 0.86 AVPR1B (0.51) GHSRF11
SCHEMBL7495104 0.86 CYP2D6 (0.50) GHSRCYP2D6ABCC1HTR2CKCNH2
SCHEMBL5877069 0.86 F11 (0.49) GHSRCYP2D6ABCC1HTR2CKCNH2
SCHEMBL5877695 0.86 AVPR1B (0.46) GHSRABCC1KCNH2ADRA1AHRH3
SCHEMBL5876981 0.85 F11 (0.52) GHSRCYP2D6ABCC1KCNH2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060706-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-06-13 US claimed
US-7060706-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed
EP-1216233-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023364-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed