SCHEMBL5877695

SCHEMBL5877695

COc1ccc2nc(-c3cccc(C)c3)n(CC3CCCC(CN)C3)c(=O)c2c1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AVPR1B P47901 12/20 0.46
F11 P03951 1/20 0.44
GHSR Q92847 2/20 0.44
NPSR1 Q6W5P4 2/20 0.43
ADRA1A P35348 1/20 0.43
KCNH2 Q12809 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
HTT P42858 1/20 0.42
PTGER4 P35408 1/20 0.42
ABCC1 P33527 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5877712 0.95 AVPR1B (0.51) AVPR1BF11GHSR
SCHEMBL5877862 0.94 AVPR1B (0.46) AVPR1BNPSR1LMNAMAPTHTT
SCHEMBL5877978 0.94 AVPR1B (0.49) AVPR1BF11GHSRADRA1AKCNH2
SCHEMBL5877946 0.92 AVPR1A (0.48) AVPR1B
SCHEMBL5877069 0.92 F11 (0.49) AVPR1BF11GHSRADRA1AKCNH2
SCHEMBL5877563 0.91 F11 (0.50) AVPR1BF11GHSRNPSR1ADRA1A
SCHEMBL5876981 0.91 F11 (0.52) AVPR1BF11GHSRADRA1AKCNH2
SCHEMBL5877811 0.91 ABCC1 (0.46) AVPR1BGHSRKCNH2ABCC1
SCHEMBL5877542 0.90 F11 (0.46) AVPR1BF11GHSRADRA1AKCNH2
SCHEMBL5877963 0.89 ALDH1A1 (0.47) AVPR1BF11GHSRNPSR1ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060706-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed
EP-1216233-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023364-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed