SCHEMBL587829

SCHEMBL587829

COC(=O)C1CCN(C(=O)OC)C(c2ccc(F)cc2F)C1.COC(=O)N1CCC(C(=O)O)CC1c1ccc(F)cc1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.38
DPP8 Q6V1X1 1/20 0.38
DPP9 Q86TI2 1/20 0.38
DPP7 Q9UHL4 1/20 0.38
TP53 P04637 1/20 0.38
ALDH1A1 P00352 3/20 0.38
TDP1 Q9NUW8 1/20 0.38
HTT P42858 1/20 0.37
MMP1 P03956 1/20 0.37
ADAM17 P78536 1/20 0.37
SLC6A9 P48067 4/20 0.36
P2RX7 Q99572 1/20 0.35
NOTUM Q6P988 1/20 0.35
HCRTR2 O43614 1/20 0.35
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
RAB9A P51151 1/20 0.34
OPRK1 P41145 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL586709 0.96 TP53 (0.41) DPP4DPP8DPP9DPP7TP53
SCHEMBL581326 0.96 TP53 (0.41) TP53ALDH1A1TDP1HTTSLC6A9
SCHEMBL587087 0.90 KMT2A (0.39) ALDH1A1NOTUMMEN1MAPTKMT2A
SCHEMBL587099 0.88 ALDH1A1 (0.34) DPP4DPP8DPP9DPP7TP53
SCHEMBL587216 0.85 KMT2A (0.41) DPP4DPP8DPP9DPP7ALDH1A1
SCHEMBL582067 0.85 CYP2C9 (0.41) NOTUMMAPTKMT2A
SCHEMBL580928 0.85 CYP2C19 (0.39) P2RX7NOTUMMAPTKMT2AHSD11B1
SCHEMBL587349 0.84 MMP1 (0.41) MMP1ADAM17NOTUM
Hydrochloric Acid SCHEMBL580918 0.84 DPP4 (0.34) DPP4DPP8DPP9DPP7TP53
SCHEMBL581895 0.83 NOTUM (0.33) DPP4DPP8DPP9DPP7NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed