SCHEMBL587349

SCHEMBL587349

COC(=O)C1CCN(C(=O)OC)C(c2ccc(F)cc2)C1.COC(=O)N1CCC(C(=O)O)CC1c1ccc(F)cc1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 2/20 0.41
ADAM17 P78536 2/20 0.41
SLC6A3 Q01959 10/20 0.41
SLC6A4 P31645 5/20 0.41
SLC6A2 P23975 3/20 0.41
NOTUM Q6P988 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL581784 0.95 NOTUM (0.44) SLC6A3SLC6A4SLC6A2NOTUM
SCHEMBL587352 0.95 SLC6A3 (0.44) MMP1ADAM17SLC6A3SLC6A4SLC6A2
SCHEMBL587433 0.88 SMN1; SMN2 (0.44) SLC6A3SLC6A4SLC6A2NOTUM
SCHEMBL587515 0.88 FFAR2 (0.39) MMP1ADAM17SLC6A3SLC6A4SLC6A2
SCHEMBL586674 0.88 NOTUM (0.44) NOTUM
SCHEMBL587575 0.85 SLC6A4 (0.43) MMP1ADAM17SLC6A4
SCHEMBL582040 0.85 ALDH1A1 (0.48) SLC6A3SLC6A4SLC6A2
SCHEMBL587629 0.85 ALDH1A1 (0.34) MMP1ADAM17SLC6A3SLC6A4SLC6A2
SCHEMBL587829 0.84 DPP4 (0.38) MMP1ADAM17NOTUM
SCHEMBL582155 0.84 RIPK1 (0.47) SLC6A3SLC6A4SLC6A2NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed