SCHEMBL5879802

SCHEMBL5879802

N#Cc1csc(CNC(=O)O)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 1/20 0.44
CYP1A2 P05177 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2D6 P10635 1/20 0.39
GRM1 Q13255 1/20 0.39
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
HSP90AA1 P07900 1/20 0.34
HDAC1 Q13547 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
CTSK P43235 1/20 0.32
POLB P06746 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32
SLC40A1 Q9NP59 1/20 0.31
ALOX15 P16050 1/20 0.31
SLC2A1 P11166 1/20 0.31
SLC2A3 P11169 1/20 0.31
SLC2A4 P14672 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23547599 0.86 NPSR1 (0.44) GABRA5CYP1A2CYP2C9CYP2D6GRM1
SCHEMBL23570691 0.82 GABRA5 (0.41) GABRA5CYP1A2CYP2C9CYP2D6GRM1
SCHEMBL6339332 0.79 HDAC3 (0.45) GABRA5HDAC1HDAC6CTSKLMNA
SCHEMBL30457818 0.75 HDAC6 (0.41) GABRA5CYP1A2CYP2C9CYP2D6GRM1
SCHEMBL19259693 0.75 ROCK2 (0.41) CYP1A2CYP2C9CYP2D6NPC1RAB9A
SCHEMBL29999682 0.75 NPC1 (0.36) CYP1A2CYP2C9CYP2D6NPC1RAB9A
SCHEMBL2909009 0.74 RAB9A (0.39) NPC1RAB9AHSP90AA1HDAC1HDAC6
SCHEMBL15110955 0.73
SCHEMBL2953054 0.71 NPSR1 (0.49) CYP1A2CYP2C9CYP2D6NPC1RAB9A
SCHEMBL19815098 0.70 GABRA5 (0.42) GABRA5RAB9AHDAC1HDAC6SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7125883-B1 Integrin receptor ligands ABBOTT GMBH & CO. KG (DE) 2006-10-24 US disclosed
US-7105508-B1 Integrin receptors antagonists ABBOTT GMBH & CO. KG (DE) 2006-09-12 US disclosed