SCHEMBL5885445

SCHEMBL5885445

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nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
TSHR P16473 1/20 0.41
GRIK1 P39086 1/20 0.39
GRIK2 Q13002 1/20 0.39
GRM1 Q13255 1/20 0.39
GRM2 Q14416 1/20 0.39
ALOX15 P16050 1/20 0.37
MAPT P10636 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C19 P33261 2/20 0.35
NPSR1 Q6W5P4 1/20 0.34
GLO1 Q04760 1/20 0.34
CYP2C9 P11712 1/20 0.33
LMNA P02545 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CASP1 P29466 1/20 0.33
THRB P10828 1/20 0.32
EGLN1 Q9GZT9 1/20 0.32
MGAM O43451 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1604823 1.00 ALDH1A1 (0.41) ALDH1A1TSHRGRIK1GRIK2GRM1
SCHEMBL4543582 1.00 ALDH1A1 (0.41) ALDH1A1TSHRGRIK1GRIK2GRM1
Hydrochloric Acid SCHEMBL1802512 0.98 ALDH1A1 (0.40) ALDH1A1TSHRGRIK1GRIK2GRM1
Hydrochloric Acid SCHEMBL1804048 0.98 ALDH1A1 (0.40) ALDH1A1TSHRGRIK1GRIK2GRM1
Hydrochloric Acid SCHEMBL4178709 0.98 ALDH1A1 (0.40) ALDH1A1TSHRGRIK1GRIK2GRM1
Hydrochloric Acid SCHEMBL9486353 0.87 GRIK1 (0.59) ALDH1A1TSHRGRIK1GRIK2GRM1
SCHEMBL4112630 0.85 GRIK1 (0.59) ALDH1A1TSHRGRIK1GRIK2GRM1
Hydrochloric Acid SCHEMBL1427352 0.83 GRIK1 (0.57) ALDH1A1TSHRGRIK1GRIK2GRM1
SCHEMBL15299749 0.80 ALDH1A1 (0.41) ALDH1A1TSHRGRIK1GRIK2GRM1
SCHEMBL15298839 0.80 ALDH1A1 (0.41) ALDH1A1TSHRGRIK1GRIK2GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060825-B2 Process for synthesizing 6-quinazolinyl-ethyl-benzoyl and related antifolates BIONUMERIK PHARMACEUTICALS, INC. (US) 2006-06-13 US claimed
US-7060825-B2 Process for synthesizing 6-quinazolinyl-ethyl-benzoyl and related antifolates BIONUMERIK PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed
US-20050020833-A1 Process for synthesizing antifolates BIONUMERIK PHARMACEUTICALS, INC. 2005-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050020833-A1 Process for synthesizing antifolates DHFR, FDPS, FOLR1 ALDH1A1 2024/4885TSHR 2859/4885GRIK1 2000/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.