SCHEMBL5886015

SCHEMBL5886015

CCN(Cc1ccc(NC2=NCCN2)cc1)C(=O)c1ccc(OC)cc1

nearest known ligand 0.69

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 11/20 0.69
ADRA2A P08913 7/20 0.62
ADRA2B P18089 6/20 0.62
ADRA2C P18825 6/20 0.62
GPR65 Q8IYL9 1/20 0.50
OPRM1 P35372 1/20 0.47
OPRD1 P41143 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5654971 0.88 PTGIR (0.70) PTGIRADRA2AADRA2BADRA2CGPR65
SCHEMBL5656120 0.87 ADRA2A (0.55) PTGIRADRA2AADRA2BADRA2CGPR65
SCHEMBL5658201 0.85 PTGIR (0.65) PTGIRADRA2AADRA2BADRA2CGPR65
SCHEMBL5656473 0.81 PTGIR (0.71) PTGIRADRA2AADRA2BADRA2CGPR65
SCHEMBL4686704 0.79 PTGIR (1.00) PTGIRADRA2AADRA2BADRA2CGPR65
SCHEMBL13017285 0.79 ADRA2A (1.00) PTGIRADRA2AADRA2BADRA2C
SCHEMBL5655170 0.78 PTGIR (0.67) PTGIRADRA2AADRA2BADRA2CGPR65
SCHEMBL6158355 0.78 PTGIR (0.74) PTGIRADRA2AADRA2BADRA2C
SCHEMBL5659732 0.78 PTGIR (0.70) PTGIRADRA2AADRA2BADRA2CGPR65
SCHEMBL6158402 0.76 PTGIR (0.63) PTGIRADRA2AADRA2BADRA2CGPR65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7279498-B2 Substituted aryl amides as IP antagonists ROCHE PALO ALTO LLC (US) 2007-10-09 US disclosed
US-7279498-B2 Substituted aryl amides as IP antagonists ROCHE PALO ALTO LLC (US) 2007-10-09 US disclosed
US-6998414-B2 Substituted arylamides as IP antagonists ROCHE PALO ALTO LLC (US) 2006-02-14 US disclosed