SCHEMBL5886750

SCHEMBL5886750

Cc1nc(N2CCc3ccccc3C2)nc2c1ccc(=O)n2-c1ccc(C(=O)NCc2ccccc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADAMTS4 O75173 7/20 0.45
LMNA P02545 3/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MAPT P10636 3/20 0.41
TP53 P04637 1/20 0.41
NAMPT P43490 1/20 0.40
ALDH1A1 P00352 2/20 0.39
POLB P06746 1/20 0.38
ROCK2 O75116 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5887024 0.92 MAPT (0.44) ADAMTS4LMNASMN1; SMN2MAPTTP53
SCHEMBL5886832 0.89 NAMPT (0.49) ADAMTS4LMNASMN1; SMN2MAPTNAMPT
SCHEMBL5887343 0.89 PRMT5 (0.43) ADAMTS4LMNAMAPTALDH1A1
SCHEMBL5886898 0.88 HPGD (0.45) LMNASMN1; SMN2MAPTTP53ALDH1A1
SCHEMBL5887548 0.88 KMT2A (0.46) LMNAMAPTTP53ALDH1A1POLB
SCHEMBL5886779 0.88 MAPT (0.44) LMNASMN1; SMN2MAPTTP53ALDH1A1
SCHEMBL5886891 0.87 TP53 (0.44) LMNASMN1; SMN2MAPTTP53ALDH1A1
SCHEMBL5886722 0.87 RXRA (0.46) ADAMTS4MAPTALDH1A1
Dimethylamine SCHEMBL5887448 0.86 HDAC6 (0.42) ADAMTS4LMNAMAPTNAMPTALDH1A1
SCHEMBL5887054 0.86 HDAC6 (0.46) ADAMTS4LMNAMAPTTP53NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US claimed
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors PHARMACIA ITALIA S.P.A. 2004-01-15 US claimed
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors TERT, TERF2, TERF2IP ADAMTS4 2688/4885LMNA 711/4885SMN1; SMN2 2219/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.