SCHEMBL5886955

SCHEMBL5886955

Cc1nc(NCc2ccccc2)nc2c1ccc(=O)n2-c1ccc(C(=O)NCc2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.48
TP53 P04637 1/20 0.48
ALDH1A1 P00352 4/20 0.46
LMNA P02545 3/20 0.46
RXFP1 Q9HBX9 2/20 0.43
POLB P06746 3/20 0.43
RAB9A P51151 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
KDR P35968 1/20 0.42
AKT1 P31749 2/20 0.42
MEN1 O00255 1/20 0.42
RECQL P46063 1/20 0.42
BLM P54132 1/20 0.42
KMT2A Q03164 1/20 0.42
MCL1 Q07820 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
AKT2 P31751 1/20 0.42
AKT3 Q9Y243 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5886840 0.93 MAPT (0.44) MAPTTP53ALDH1A1LMNARXFP1
SCHEMBL5886920 0.93 MAPT (0.44) MAPTTP53ALDH1A1LMNARXFP1
SCHEMBL5886935 0.92 RAB9A (0.47) MAPTTP53LMNARXFP1RAB9A
SCHEMBL5887012 0.92 MAPT (0.43) MAPTTP53ALDH1A1LMNARXFP1
SCHEMBL5886922 0.92 MAPT (0.46) MAPTTP53ALDH1A1LMNAMEN1
SCHEMBL5887676 0.92 MAPT (0.43) MAPTTP53ALDH1A1LMNARXFP1
SCHEMBL5886892 0.92 MAPT (0.41) MAPTTP53ALDH1A1LMNARXFP1
SCHEMBL5887092 0.91 MAPT (0.46) MAPTTP53ALDH1A1LMNARXFP1
SCHEMBL5886708 0.91 TP53 (0.48) MAPTTP53ALDH1A1LMNARXFP1
SCHEMBL5887041 0.90 MAPT (0.42) MAPTTP53ALDH1A1LMNARXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US claimed
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors PHARMACIA ITALIA S.P.A. 2004-01-15 US claimed
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors TERT, TERF2, TERF2IP MAPT 1614/4885TP53 43/4885ALDH1A1 1860/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.