SCHEMBL5887085

SCHEMBL5887085

Cc1nc(N2CCN(C(=O)c3cccnc3)CC2)nc2c1ccc(=O)n2-c1ccc(C(=O)NCc2ccc(C(=O)O)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.41
MAPT P10636 2/20 0.41
KLKB1 P03952 1/20 0.40
KLK1 P06870 1/20 0.40
KHK P50053 1/20 0.40
NAMPT P43490 3/20 0.40
MYC P01106 1/20 0.40
AKT1 P31749 2/20 0.39
AKT2 P31751 2/20 0.39
AKT3 Q9Y243 2/20 0.39
MMP12 P39900 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5887048 0.96 MAPT (0.42) HTTMAPTKLKB1KLK1KHK
SCHEMBL5887505 0.93 MGAM (0.41) HTTMAPTKLKB1KLK1KHK
SCHEMBL5887563 0.92 EPHX2 (0.42) HTTMAPTNAMPTHDAC3HDAC4
SCHEMBL5887646 0.92 MAPK1 (0.40) HTTMAPTKLKB1KLK1NAMPT
SCHEMBL5887334 0.89 ALDH1A1 (0.44) HTTMAPTNAMPTGAAMEN1
SCHEMBL5887675 0.89 SLC6A7 (0.44) MAPTKLKB1MEN1KMT2AALDH1A1
SCHEMBL5886700 0.86 MGLL (0.42) MAPTKLKB1MEN1KMT2AALDH1A1
SCHEMBL5887572 0.85 MAPT (0.39) HTTMAPTKLKB1KHKMMP12
SCHEMBL5886889 0.85 MAPK10 (0.45) NAMPTMEN1KMT2ASMN1; SMN2
SCHEMBL5886777 0.85 NAMPT (0.46) HTTMAPTNAMPTHDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US disclosed