SCHEMBL5887244

SCHEMBL5887244

Cc1nc(Oc2ccc(F)cc2)nc2c1ccc(=O)n2-c1ccc(C(=O)NC2CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 5/20 0.44
PDE4B Q07343 1/20 0.41
PDE4D Q08499 1/20 0.41
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
CCNE1 P24864 3/20 0.40
CDK2 P24941 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
TTK P33981 1/20 0.40
MCHR1 Q99705 2/20 0.40
MAPK8 P45983 1/20 0.40
THRB P10828 1/20 0.40
ADRA2A P08913 1/20 0.39
ADRA1A P35348 1/20 0.39
HRH1 P35367 1/20 0.39
HTR2B P41595 1/20 0.39
HPGD P15428 2/20 0.39
CDK4 P11802 1/20 0.39
CCND1 P24385 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5887013 0.92 TTK (0.40) MAPK14PDE4BNPC1RAB9ATTK
SCHEMBL5886782 0.91 PDE4B (0.44) PDE4BTTKMCHR1MAPK8THRB
SCHEMBL5887588 0.89 SMN1; SMN2 (0.42) MAPK14PDE4BKMT2AMEN1TTK
SCHEMBL5887451 0.87 MAPK8 (0.42) PDE4BTTKMAPK8THRBALDH1A1
SCHEMBL5887445 0.87 KMT2A (0.38) PDE4BKMT2AMEN1TTKMAPK8
SCHEMBL5887052 0.84 PARP10 (0.39) MAPK14KMT2AMEN1HPGDALDH1A1
SCHEMBL5887651 0.82 PDE4B (0.41) MAPK14PDE4BPDE4DKMT2ACCNE1
SCHEMBL5887152 0.82 CCNE1 (0.48) PDE4BPDE4DCCNE1CDK2NPC1
SCHEMBL5886789 0.82 HPGD (0.47) MAPK14KMT2AMEN1MAPK8HPGD
SCHEMBL5887454 0.81 PDE4B (0.38) MAPK14PDE4BPDE4DTTKMAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US claimed
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors PHARMACIA ITALIA S.P.A. 2004-01-15 US claimed
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors TERT, TERF2, TERF2IP MAPK14 1051/4885PDE4B 2197/4885PDE4D 2134/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.