SCHEMBL5887377

SCHEMBL5887377

CCOc1cccc(C2=CC(OC)=CC[CH]2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.42
GAA P10253 2/20 0.42
KDM4E B2RXH2 2/20 0.42
RXRA P19793 1/20 0.42
RXRB P28702 1/20 0.42
THRB P10828 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
TP53 P04637 2/20 0.41
CYP3A4 P08684 1/20 0.41
BRD4 O60885 1/20 0.40
BRD2 P25440 1/20 0.40
CREBBP Q92793 1/20 0.40
NOTUM Q6P988 1/20 0.40
FGFR1 P11362 1/20 0.39
FGFR2 P21802 1/20 0.39
FGFR3 P22607 1/20 0.39
ALDH1A1 P00352 2/20 0.38
TSHR P16473 2/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5887546 0.87 DYRK1A (0.44) GAACYP3A4NOTUMCYP1A2CYP2D6
SCHEMBL4804654 0.78 ACHE (0.39) KDM4ETDP1TP53ALDH1A1TSHR
SCHEMBL6408167 0.77 MAPT (0.33) MAPTKDM4ETP53ALDH1A1TSHR
SCHEMBL6047594 0.77 NAAA (0.40) MAPTKDM4ERXRARXRBTHRB
SCHEMBL4012746 0.74 NOTUM (0.36) MAPTKDM4ETP53NOTUMALDH1A1
SCHEMBL6047605 0.74 CYP1A1 (0.44) THRBCYP3A4BRD4ALDH1A1LMNA
SCHEMBL5887031 0.73 CDC25A (0.44) GAATDP1RAB9ANPC1DHFR
SCHEMBL29426410 0.73 RXRA (0.66) MAPTGAAKDM4ERXRARXRB
SCHEMBL9260410 0.73 RXRA (0.66) MAPTGAAKDM4ERXRARXRB
SCHEMBL29012837 0.71 RXRA (0.64) MAPTGAAKDM4ERXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7037931-B2 Corticotropin releasing factor moderator; analgesics; drug abruse, drug dependency; schizophrenia JANSSEN PHARMACEUTICA N.V. (BE) 2006-05-02 US claimed