SCHEMBL5887580

SCHEMBL5887580

Cc1ccc(C2=C(c3cccc(Cl)c3)[CH]CC=C2C(F)(F)F)cc1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
HSD17B1 P14061 1/20 0.32
HSD17B2 P37059 1/20 0.32
DHODH Q02127 1/20 0.32
PDK2 Q15119 1/20 0.32
PGR P06401 2/20 0.32
PTGS2 P35354 1/20 0.31
ALOX5 P09917 1/20 0.31
PTPN5 P54829 1/20 0.31
TAAR1 Q96RJ0 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5887149 0.88 AR (0.38) HSD17B1HSD17B2PDK2PTGS2PTPN5
SCHEMBL5887499 0.83 ALKBH3 (0.41) SMN1; SMN2HSD17B1HSD17B2PGR
SCHEMBL5887236 0.82 ESR2 (0.35) ESR2SMN1; SMN2PDK2PGRPTGS2
SCHEMBL5887105 0.79 ESR2 (0.35) ESR2SMN1; SMN2ALOX5
SCHEMBL5887498 0.79 HSD11B1 (0.34) PDK2
SCHEMBL4808757 0.75 ESR2 (0.39) ESR2SMN1; SMN2PGRALOX5TAAR1
SCHEMBL4012821 0.72 ESR2 (0.36) ESR2SMN1; SMN2ALOX5
SCHEMBL5887155 0.70 NOTUM (0.36) ESR2SMN1; SMN2ALOX5TAAR1
SCHEMBL4013100 0.69 ESR2 (0.39) ESR2SMN1; SMN2PGRALOX5TAAR1
SCHEMBL6047606 0.69 NR1I3 (0.39) SMN1; SMN2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7037931-B2 Corticotropin releasing factor moderator; analgesics; drug abruse, drug dependency; schizophrenia JANSSEN PHARMACEUTICA N.V. (BE) 2006-05-02 US claimed