SCHEMBL5887498

SCHEMBL5887498

Cc1ccc(C2=C(c3ccccc3Cl)[CH]CC=C2C(F)(F)F)cc1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
AR P10275 1/20 0.33
PDK2 Q15119 3/20 0.31
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
HPGD P15428 1/20 0.30
ALOX15 P16050 1/20 0.30
CYP2C19 P33261 1/20 0.30
HSD17B10 Q99714 1/20 0.30
CYP2A6 P11509 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5887580 0.79 ESR2 (0.35) PDK2
SCHEMBL5887426 0.78 MEN1 (0.34) MEN1POLBKMT2ACYP2D6CYP2C9
SCHEMBL5887149 0.76 AR (0.38) MEN1KMT2AARPDK2
SCHEMBL5887499 0.72 ALKBH3 (0.41) ARCYP2C9HPGDALOX15CYP2C19
SCHEMBL5887625 0.68 HSP90AA1 (0.36) MEN1KMT2AHSD17B10CYP2A6
SCHEMBL1045000 0.66 CYP2A6 (0.65) HSD11B1MEN1POLBKMT2AHPGD
SCHEMBL5887436 0.65 CYP2A6 (0.36) HSD11B1MEN1POLBKMT2ACYP2D6
SCHEMBL5887191 0.65 MEN1 (0.37) MEN1POLBKMT2A
SCHEMBL5887347 0.64 MEN1 (0.35) MEN1POLBKMT2A
SCHEMBL6047646 0.63 CYP2D6 (0.32) CYP2D6CYP2C9HPGDALOX15CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7037931-B2 Corticotropin releasing factor moderator; analgesics; drug abruse, drug dependency; schizophrenia JANSSEN PHARMACEUTICA N.V. (BE) 2006-05-02 US claimed