SCHEMBL5887149

SCHEMBL5887149

Cc1ccc(C2=C(c3cccc(C)c3)[CH]CC=C2C(F)(F)F)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.38
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HSD17B1 P14061 1/20 0.34
HSD17B2 P37059 1/20 0.34
PTPN5 P54829 2/20 0.33
PDK2 Q15119 1/20 0.33
ENPP1 P22413 1/20 0.32
SDHB P21912 1/20 0.32
PTGS1 P23219 2/20 0.31
ORAI1 Q96D31 1/20 0.31
FYN P06241 1/20 0.30
CLK4 Q9HAZ1 1/20 0.30
DYRK1B Q9Y463 1/20 0.30
NISCH Q9Y2I1 1/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30
NFE2L2 Q16236 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5887580 0.88 ESR2 (0.35) HSD17B1HSD17B2PTPN5PDK2PTGS2
SCHEMBL5887499 0.86 ALKBH3 (0.41) ARL3MBTL1HSD17B1HSD17B2
SCHEMBL5887311 0.79 KMT2A (0.36) MEN1KMT2AL3MBTL1HSD17B1HSD17B2
SCHEMBL5887353 0.77 MEN1 (0.35) MEN1KMT2AL3MBTL1HSD17B2FYN
SCHEMBL5887498 0.76 HSD11B1 (0.34) ARMEN1KMT2APDK2
SCHEMBL5887236 0.70 ESR2 (0.35) PTPN5PDK2PTGS2
SCHEMBL5887199 0.68 KMT2A (0.35) MEN1KMT2AL3MBTL1
SCHEMBL5887285 0.67 ALKBH3 (0.44) MEN1KMT2AL3MBTL1CLK4NISCH
SCHEMBL6047649 0.66 L3MBTL1 (0.38) MEN1KMT2AL3MBTL1NISCHCHRNB4
SCHEMBL5887245 0.66 AR (0.31) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7037931-B2 Corticotropin releasing factor moderator; analgesics; drug abruse, drug dependency; schizophrenia JANSSEN PHARMACEUTICA N.V. (BE) 2006-05-02 US claimed