SCHEMBL5889555

SCHEMBL5889555

CCCn1c(C(=O)NCCN)cc2cc(NC(=O)c3ccc4[nH]c(C(=O)Nc5ccc6c(c5)cc(C(=O)NCCN)n6CCC)cc4c3)ccc21

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRAS P01112 3/20 0.47
ESR1 P03372 3/20 0.47
ESR2 Q92731 3/20 0.47
HDAC2 Q92769 2/20 0.44
ROCK2 O75116 1/20 0.42
PLD2 O14939 1/20 0.41
PLD1 Q13393 1/20 0.41
ITGB3 P05106 10/20 0.41
ITGA2B P08514 10/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
KDM4E B2RXH2 1/20 0.39
NHERF1 O14745 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5889686 0.97 HRAS (0.45) HRASESR1ESR2HDAC2ROCK2
SCHEMBL6500730 0.89 HRAS (0.44) HRASESR1ESR2HDAC2ROCK2
SCHEMBL5677265 0.81 ITGB3 (0.54) HDAC2PLD2PLD1ITGB3ITGA2B
SCHEMBL5889571 0.80 HRAS (0.59) HRASESR1ESR2HDAC2ROCK2
SCHEMBL5889689 0.79 NPC1 (0.46) HRASESR1ESR2HDAC2ROCK2
SCHEMBL5680312 0.78 NHERF1 (0.54) HDAC2PLD2PLD1ITGB3ITGA2B
SCHEMBL5889537 0.78 KDM4E (0.51) HDAC2PLD2PLD1ITGB3ITGA2B
SCHEMBL5679912 0.77 MMP13 (0.62) HDAC2PLD2PLD1ITGB3ITGA2B
SCHEMBL5896655 0.76 KDM4E (0.51) HDAC2PLD2PLD1ITGB3ITGA2B
SCHEMBL5889562 0.76 HDAC2 (0.50) HDAC2ROCK2ITGB3ITGA2BKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7064218-B2 Aromatic compounds and poly(oxyalkylene) containing aromatic compounds possessing antibacterial, antifungal or antitumor activity GENELABS TECHNOLOGIES, INC. (US) 2006-06-20 US disclosed
US-20030212113-A1 Novel aromatic compounds and poly(oxyalkylene) containing aromatic compounds possessing antibacterial, antifungal or antitumor activity GLAXOSMITHKLINE LLC 2003-11-13 US disclosed
WO-2003057212-A1 POLYAMIDE DERIVATIVES POSSESSING ANTIBACTERIAL, ANTIFUNGAL OR ANTITUMOR ACTIVITY GENELABS TECHNOLOGIES, INC. (US) 2003-07-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030212113-A1 Novel aromatic compounds and poly(oxyalkylene) containing aromatic compounds possessing antibacterial, antifungal or antitumor activity TYR, CYP51A1, ODC1 HRAS 1040/4885ESR1 4541/4885ESR2 4085/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.