SCHEMBL5897283

SCHEMBL5897283

COc1ccc(C(CC(=O)NCc2ccc(NC(=O)Nc3ccccc3C)cc2)NC(=O)c2ccc(C(=O)OC(C)(C)C)cc2)cc1OC

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 8/20 0.53
ITGA4 P13612 8/20 0.53
MAPT P10636 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
NAMPT P43490 4/20 0.42
ITGB7 P26010 1/20 0.42
HDAC1 Q13547 3/20 0.41
HDAC2 Q92769 2/20 0.41
HDAC11 Q96DB2 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
MEN1 O00255 1/20 0.40
GAA P10253 1/20 0.40
KMT2A Q03164 1/20 0.40
P2RX7 Q99572 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5896459 0.93 ITGB1 (0.53) ITGB1ITGA4MAPTNPC1RAB9A
SCHEMBL5865240 0.90 ITGB1 (0.58) ITGB1ITGA4MAPTNPC1RAB9A
SCHEMBL5897280 0.86 ITGB1 (0.53) ITGB1ITGA4MAPTNAMPTITGB7
SCHEMBL5896625 0.82 ITGB1 (0.58) ITGB1ITGA4MAPTNPC1RAB9A
SCHEMBL6353998 0.80 ITGB1 (0.61) ITGB1ITGA4ITGB7
SCHEMBL5896454 0.79 ITGB1 (0.53) ITGB1ITGA4MAPTNPC1RAB9A
SCHEMBL6344233 0.78 ITGB1 (0.59) ITGB1ITGA4ITGB7
SCHEMBL5700782 0.75 ITGB1 (0.65) ITGB1ITGA4ITGB7MEN1KMT2A
SCHEMBL5897049 0.74 POLB (0.54) MAPTKMT2A
SCHEMBL5896878 0.73 MAPT (0.47) MAPTNPC1MEN1GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7091242-B2 Beta-amino acid derivatives as integrin receptor antagonists BAYER AKTIENGESELLSCHAFT (DE) 2006-08-15 US disclosed