2-Picolinic Acid

2-Picolinic Acid

SCHEMBL593180

O=C(O)c1ccccn1.O=C(O)c1ccccn1.O=C(O)c1ccccn1.O=C([O-])c1cc(O)ccn1.O=C([O-])c1cc(O)ccn1.O=C([O-])c1cc(O)ccn1.[Eu+3]

nearest known ligand 0.61

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.61
L3MBTL1 Q9Y468 2/20 0.61
NAPRT Q6XQN6 1/20 0.61
P4HTM Q9NXG6 1/20 0.61
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
KMT2A Q03164 1/20 0.44
ALDH1A1 P00352 4/20 0.42
KDM4E B2RXH2 5/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
OPRK1 P41145 1/20 0.41
HTT P42858 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KDM5A P29375 2/20 0.41
KDM6B O15054 2/20 0.41
KDM4A O75164 2/20 0.41
KDM5C P41229 2/20 0.41
KDM4C Q9H3R0 2/20 0.41
KDM2A Q9Y2K7 2/20 0.41
KDM3A Q9Y4C1 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
2-Picolinic Acid SCHEMBL594569 0.97 LMNA (0.61) LMNAL3MBTL1NAPRTP4HTMCES2
2-Picolinic Acid SCHEMBL12076591 0.97 LMNA (0.61) LMNAL3MBTL1NAPRTP4HTMCES2
2-Picolinic Acid SCHEMBL593292 0.94 LMNA (0.56) LMNAL3MBTL1NAPRTP4HTMCES2
2-Picolinic Acid SCHEMBL593739 0.91 LMNA (0.56) LMNAL3MBTL1NAPRTP4HTMCES2
SCHEMBL2362971 0.89 KDM4E (0.52) LMNAL3MBTL1NAPRTP4HTMALDH1A1
2-Picolinic Acid SCHEMBL595042 0.87 LMNA (0.69) LMNAL3MBTL1NAPRTP4HTMCES2
2-Picolinic Acid SCHEMBL593726 0.87 LMNA (0.69) LMNAL3MBTL1NAPRTP4HTMCES2
SCHEMBL29951101 0.78 KDM4E (0.63) LMNAL3MBTL1NAPRTP4HTMALDH1A1
2-Picolinic Acid SCHEMBL28737738 0.78 CES2 (0.64) LMNAL3MBTL1NAPRTP4HTMCES2
SCHEMBL65841 0.78 KDM4E (0.63) LMNAL3MBTL1NAPRTP4HTMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2294159-B1 DISTANCE-CONTROLLED ENERGY TRANSFER DYE COMPLEXES INBIO PROF JUERGEN BUEDDEFELD DR PETER KLAUTH PROF MANFRED RIETZ GBR (DE) 2012-09-05 EP claimed
US-20110189781-A1 DISTANCE-CONTROLLED ENERGY TRANSFER DYE COMPLEXES BÜDDEFELD, JÜRGEN, PROF (DE) 2011-08-04 US claimed
EP-2294159-B1 DISTANCE-CONTROLLED ENERGY TRANSFER DYE COMPLEXES INBIO PROF JUERGEN BUEDDEFELD DR PETER KLAUTH PROF MANFRED RIETZ GBR (DE) 2012-09-05 EP disclosed
EP-2417216-A2 MODIFICATION OF LAYERED SILICATES FOR LUMINESCENCE ACTIVATION Inbio Prof. Jürgen Büddefeld Dr. Peter Klauth Prof. Manfred Rietz Gbr (DE) 2012-02-15 EP disclosed
US-20110189781-A1 DISTANCE-CONTROLLED ENERGY TRANSFER DYE COMPLEXES BÜDDEFELD, JÜRGEN, PROF (DE) 2011-08-04 US disclosed
WO-2010115503-A2 MODIFICATION OF LAYERED SILICATES FOR LUMINESCENCE ACTIVATION INBIO PROF. JÜRGEN BÜDDEFELD DR. PETER KLAUTH PROF. MANFRED RIETZ GBR (DE) 2010-10-14 WO disclosed