SCHEMBL594177

SCHEMBL594177

O=C(O)c1cc2ccccc2cc1-c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.57
GPR35 Q9HC97 2/20 0.53
PTPN1 P18031 3/20 0.52
ALDH1A1 P00352 2/20 0.52
KDM4E B2RXH2 1/20 0.52
HPGD P15428 1/20 0.52
MYC P01106 1/20 0.51
FOLH1 Q04609 1/20 0.51
MAPT P10636 2/20 0.50
GFER P55789 1/20 0.50
NGLY1 Q96IV0 1/20 0.50
HNF4A P41235 1/20 0.50
AKR1C3 P42330 1/20 0.49
AKR1C2 P52895 1/20 0.49
AKR1C1 Q04828 1/20 0.49
ACMSD Q8TDX5 1/20 0.49
GPR84 Q9NQS5 1/20 0.47
PTPN2 P17706 1/20 0.47
PTPN6 P29350 1/20 0.47
ALOX15 P16050 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL667582 0.87 PTPN1 (0.59) PTPN1ALDH1A1FOLH1HNF4AAKR1C3
SCHEMBL27542885 0.86 ACMSD (0.62) IDO1ALDH1A1KDM4EHPGDMYC
SCHEMBL9171492 0.85 PTPN1 (0.57) PTPN1ALDH1A1FOLH1HNF4AAKR1C3
SCHEMBL10058716 0.84 MYC (0.50) IDO1ALDH1A1KDM4EHPGDMYC
SCHEMBL28052572 0.84 PTGS2 (0.47) IDO1GPR35PTPN1ALDH1A1KDM4E
SCHEMBL613285 0.83 BACE1 (0.50) IDO1ALDH1A1KDM4EHPGDMAPT
SCHEMBL14034445 0.83 FOLH1 (0.53) IDO1GPR35PTPN1FOLH1HNF4A
SCHEMBL5569233 0.83 PTPN1 (0.55) PTPN1ALDH1A1FOLH1HNF4AAKR1C3
SCHEMBL28439181 0.83 PTPN1 (0.55) PTPN1ALDH1A1FOLH1HNF4AAKR1C3
SCHEMBL69178 0.82 IDO1 (0.71) IDO1GPR35PTPN1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115057776-B Synthesis method of ethyl 2-naphthoate derivative 必维申瓯质量技术服务温州有限公司 2023-08-22 CN disclosed
US-8114993-B2 Use of aryl chlorides in palladium-catalyzed C-H bond functionalization THE UNIVERSITY OF HOUSTON SYSTEM (US) 2012-02-14 US disclosed
US-8114993-B2 Use of aryl chlorides in palladium-catalyzed C-H bond functionalization THE UNIVERSITY OF HOUSTON SYSTEM (US) 2012-02-14 US disclosed
US-8114993-B2 Use of aryl chlorides in palladium-catalyzed C-H bond functionalization THE UNIVERSITY OF HOUSTON SYSTEM (US) 2012-02-14 US disclosed
US-20090012293-A1 USE OF ARYL CHLORIDES IN PALLADIUM-CATALYZED C-H BOND FUNCTIONALIZATION THE UNIVERSITY OF HOUSTON SYSTEM (US) 2009-01-08 US disclosed
US-20090012293-A1 USE OF ARYL CHLORIDES IN PALLADIUM-CATALYZED C-H BOND FUNCTIONALIZATION THE UNIVERSITY OF HOUSTON SYSTEM (US) 2009-01-08 US disclosed
US-20090012293-A1 USE OF ARYL CHLORIDES IN PALLADIUM-CATALYZED C-H BOND FUNCTIONALIZATION THE UNIVERSITY OF HOUSTON SYSTEM (US) 2009-01-08 US disclosed
EP-1091958-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2001-04-18 EP disclosed
WO-2000001692-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2000-01-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090012293-A1 USE OF ARYL CHLORIDES IN PALLADIUM-CATALYZED C-H BOND FUNCTIONALIZATION DBH, DDT, CYCS IDO1 522/4885GPR35 1633/4885PTPN1 3231/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.