SCHEMBL5951850

SCHEMBL5951850

COC(=O)c1cccc(-c2cccc3c2C(=O)C(C)C3)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.44
CA9 Q16790 2/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
ERN1 O75460 2/20 0.43
ACHE P22303 2/20 0.42
CHRM2 P08172 1/20 0.41
CHRM4 P08173 1/20 0.41
CHRM5 P08912 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
FOLH1 Q04609 1/20 0.41
MGAT2 Q10469 1/20 0.41
DGAT2 Q96PD7 1/20 0.41
HCRTR1 O43613 1/20 0.41
HCRTR2 O43614 1/20 0.41
PDK2 Q15119 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
AXL P30530 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5952849 0.88 EGFR (0.45) CA12CA9CA1CA2ACHE
SCHEMBL5951324 0.82 ACHE (0.52) CA12CA9CA1CA2ERN1
SCHEMBL5952665 0.80 ACHE (0.54) ACHEALDH1A1LMNA
SCHEMBL5951226 0.79 TDP2 (0.52) ACHE
SCHEMBL5952024 0.79 ACHE (0.49) ACHEPDK2ALDH1A1LMNA
SCHEMBL5951968 0.78 ACHE (0.54) ACHEHCRTR1HCRTR2
SCHEMBL5952266 0.78 ACHE (0.50) ACHENPC1RAB9AALDH1A1
SCHEMBL5509273 0.77 ACHE (0.61) ACHE
SCHEMBL5952829 0.77 ACHE (0.49) ACHE
Dimethylamine SCHEMBL7161154 0.76 ACHE (0.56) ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7038070-B2 Preparation of preparing substituted indanones BASELL POLYOLEFINE GMBH (DE) 2006-05-02 US disclosed
US-6963017-B2 Preparation of preparing substituted indanones BASELL POLYOLEFINE GMBH (DE) 2005-11-08 US disclosed
EP-0968158-B1 METHOD OF PREPARING SUBSTITUTED INDANONES, THE SUBSTITUTED INDANONES AND METALLOCENES PREPARED THEREFROM BASELL POLYOLEFINE GMBH (DE) 2005-08-10 EP disclosed
US-20050033076-A1 Preparation of preparing substituted indanones EQUISTAR CHEMICALS, LP 2005-02-10 US disclosed
US-20030009046-A1 Preparation of preparing substituted indanones EQUISTAR CHEMICALS, LP 2003-01-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050033076-A1 Preparation of preparing substituted indanones CYP1A2, CYP2J2, IDH3A CA12 3977/4885CA9 3552/4885CA1 3547/4885
US-20030009046-A1 Preparation of preparing substituted indanones CYP1A2, CYP1B1, CYP1A1 CA12 3969/4885CA9 3446/4885CA1 3105/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.