SCHEMBL5953230

SCHEMBL5953230

Cc1ccc(Cl)c2c1CC(C(F)(F)F)C2=O

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.35
MAOA P21397 4/20 0.34
MAOB P27338 2/20 0.34
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
POLL Q9UGP5 1/20 0.33
ACHE P22303 1/20 0.32
ACACB O00763 1/20 0.31
ACACA Q13085 1/20 0.31
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1023191 0.77 ACHE (0.50) CES1MAOAMAOBHTR2AHTR2C
SCHEMBL1022897 0.73 MAOA (0.42) CES1MAOAMAOBHTR2AHTR2C
SCHEMBL5952939 0.71 HTR2A (0.40) CES1HTR2AHTR2CHTR2B
SCHEMBL5952927 0.68 METAP1 (0.37) CES1ACHE
SCHEMBL5952089 0.64 ACHE (0.49) CES1MAOAHTR2CACHE
SCHEMBL8218376 0.62 CES1 (0.44) CES1MAOAMAOBHTR2AHTR2C
SCHEMBL31693572 0.61 ACHE (0.56) MAOAMAOBPOLLACHE
SCHEMBL2046109 0.61 ACHE (0.56) MAOAMAOBPOLLACHE
SCHEMBL16290540 0.60 ALDH1A1 (0.31)
SCHEMBL18264394 0.60 MAOA (0.40) MAOAMAOBPOLLACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7038070-B2 Preparation of preparing substituted indanones BASELL POLYOLEFINE GMBH (DE) 2006-05-02 US disclosed
US-6963017-B2 Preparation of preparing substituted indanones BASELL POLYOLEFINE GMBH (DE) 2005-11-08 US disclosed
EP-0968158-B1 METHOD OF PREPARING SUBSTITUTED INDANONES, THE SUBSTITUTED INDANONES AND METALLOCENES PREPARED THEREFROM BASELL POLYOLEFINE GMBH (DE) 2005-08-10 EP disclosed
US-20050033076-A1 Preparation of preparing substituted indanones EQUISTAR CHEMICALS, LP 2005-02-10 US disclosed
US-20030009046-A1 Preparation of preparing substituted indanones EQUISTAR CHEMICALS, LP 2003-01-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050033076-A1 Preparation of preparing substituted indanones CYP1A2, CYP2J2, IDH3A CES1 3217/4885MAOA 498/4885MAOB 334/4885
US-20030009046-A1 Preparation of preparing substituted indanones CYP1A2, CYP1B1, CYP1A1 CES1 2736/4885MAOA 564/4885MAOB 403/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.