SCHEMBL5960274

SCHEMBL5960274

CC(=O)c1ccc2[nH]c(C)c(C(=O)OC(C)(C)C)c2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 6/20 0.52
GABRG2 P18507 6/20 0.52
GABRB3 P28472 6/20 0.52
GABRA3 P34903 6/20 0.52
GABRA2 P47869 6/20 0.52
GAA P10253 1/20 0.48
KIF11 P52732 2/20 0.48
HCRTR1 O43613 2/20 0.46
KDM4E B2RXH2 4/20 0.44
ALDH1A1 P00352 4/20 0.44
HPGD P15428 3/20 0.44
THRB P10828 1/20 0.44
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
NR4A2 P43354 1/20 0.43
GABRA5 P31644 4/20 0.41
GABRA4 P48169 3/20 0.41
GABRA6 Q16445 3/20 0.41
HSD17B10 Q99714 2/20 0.40
MAPT P10636 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17203149 0.89 KDM4E (0.58) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL17205786 0.88 RAB9A (0.59) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL7815779 0.83 GAA (0.68) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL5960232 0.82 GAA (0.49) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL7356882 0.82 GAA (0.49) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL15174105 0.79 NR4A2 (0.69) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL9953449 0.77 KIF11 (0.49) GAAKIF11HCRTR1KDM4EALDH1A1
SCHEMBL5235955 0.76 MAPT (0.43) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL19211784 0.75 KIF11 (0.56) KIF11HCRTR1KDM4EALDH1A1HPGD
SCHEMBL14211006 0.75 KDM4E (0.75) KIF11HCRTR1KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682553-A1 THIENOPYRAZOLES Aventis Pharmaceuticals Inc. (US) 2006-07-26 EP disclosed
WO-2005026175-A1 THIENOPYRAZOLES AVENTIS PHARMACEUTICALS INC. (US) 2005-03-24 WO disclosed