SCHEMBL5960313

SCHEMBL5960313

CC(=O)c1ccc2[nH]cc(C(=O)OC(C)(C)C)c2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
ALDH1A1 P00352 1/20 0.50
TP53 P04637 1/20 0.50
HPGD P15428 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
NR4A2 P43354 7/20 0.49
HTR1A P08908 1/20 0.49
HTR1D P28221 1/20 0.49
HTR1B P28222 1/20 0.49
GABRA1 P14867 1/20 0.47
GABRG2 P18507 1/20 0.47
GABRB3 P28472 1/20 0.47
GABRA3 P34903 1/20 0.47
GABRA2 P47869 1/20 0.47
KDM4E B2RXH2 1/20 0.43
CREBBP Q92793 1/20 0.42
PBRM1 Q86U86 1/20 0.42
F7 P08709 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3930534 0.89 HSD17B10 (0.56) HSD17B10MEN1KMT2AALDH1A1TP53
SCHEMBL6630345 0.89 NR4A2 (0.49) HSD17B10MEN1KMT2AALDH1A1TP53
SCHEMBL27853728 0.88 NR4A2 (0.58) HSD17B10MEN1KMT2AALDH1A1TP53
SCHEMBL6629905 0.85 NR4A2 (0.46) HSD17B10MEN1KMT2AALDH1A1TP53
SCHEMBL28371975 0.85 NR4A2 (0.62) HSD17B10MEN1KMT2AALDH1A1TP53
SCHEMBL27909264 0.84 GABRA1 (0.54) HSD17B10MEN1KMT2AALDH1A1TP53
SCHEMBL10397437 0.84 NR4A2 (0.68) HSD17B10MEN1KMT2AALDH1A1TP53
SCHEMBL6991795 0.83 NR4A2 (0.51) ALDH1A1HPGDNR4A2KDM4ECREBBP
SCHEMBL27548934 0.82 PBRM1 (0.61) HSD17B10MEN1KMT2AALDH1A1TP53
SCHEMBL1007089 0.82 NR4A2 (0.50) MEN1KMT2AHPGDNR4A2CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682553-A1 THIENOPYRAZOLES Aventis Pharmaceuticals Inc. (US) 2006-07-26 EP disclosed
WO-2005026175-A1 THIENOPYRAZOLES AVENTIS PHARMACEUTICALS INC. (US) 2005-03-24 WO disclosed