SCHEMBL5963637

SCHEMBL5963637

O=C(O)c1oc(Br)c(Br)c1-c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
PTPN1 P18031 2/20 0.39
FABP4 P15090 1/20 0.37
GRIA4 P48058 1/20 0.37
ALDH1A1 P00352 3/20 0.37
HPGD P15428 2/20 0.37
LMNA P02545 2/20 0.36
KDM4E B2RXH2 2/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
AKR1C3 P42330 2/20 0.35
AKR1C2 P52895 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3973139 0.87 PTPN1 (0.40) NPC1RAB9APTPN1FABP4GRIA4
SCHEMBL71486 0.80 PTPN1 (0.46) NPC1RAB9APTPN1ALDH1A1HPGD
SCHEMBL3978711 0.73 PTPN1 (0.49) NPC1RAB9APTPN1ALDH1A1HPGD
SCHEMBL3977576 0.73 PTPN1 (0.41) NPC1RAB9APTPN1ALDH1A1HPGD
SCHEMBL28130850 0.72 PTPN1 (0.47) NPC1RAB9APTPN1ALDH1A1HPGD
SCHEMBL8861328 0.70 FABP4 (0.41) PTPN1FABP4ALDH1A1HPGDLMNA
SCHEMBL3610930 0.70 PTPN1 (0.59) NPC1PTPN1ALDH1A1HPGDLMNA
SCHEMBL3974214 0.69 PTGS1 (0.48) RAB9AALDH1A1HPGDLMNAKDM4E
SCHEMBL3361896 0.69 ALDH1A1 (0.61) ALDH1A1HPGDLMNAKDM4EGAA
SCHEMBL4711778 0.68 ALDH1A1 (0.46) NPC1RAB9AALDH1A1HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1143959-B1 ANTIFUNGAL ACTIVITY OF DICATIONIC MOLECULES UNIV NORTH CAROLINA (US) 2006-11-02 EP disclosed
EP-1685836-A2 Antifungal activity of dicationic molecules UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2006-08-02 EP disclosed
EP-0792271-B1 FURAN DERIVATIVES FOR INHIBITING PNEUMOCYSTIS CARINII PNEUMONIA, GIARDIA LAMBLIA AND CRYPTOSPORIDIUM PARVUM UNIV GEORGIA STATE RES FOUND (US) 2002-02-27 EP disclosed
US-6326395-B1 AMIDINE OR AMIDE SUBSTITUTED FURAN DERIVATIVES DUKE UNIVERSITY 2001-12-04 US disclosed
EP-1143959-A2 ANTIFUNGAL ACTIVITY OF DICATIONIC MOLECULES UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2001-10-17 EP disclosed
WO-2000015212-A2 ANTIFUNGAL ACTIVITY OF DICATIONIC MOLECULES THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2000-03-23 WO disclosed
US-5602172-A USING A 2,5-DIPHENYLFURAN COMPOUND THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1997-02-11 US disclosed