SCHEMBL597398

SCHEMBL597398

CCC(C(=O)O)c1c(C)[nH]c2cccc(Br)c12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR17 Q13304 1/20 0.41
FEN1 P39748 1/20 0.38
MAPT P10636 4/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
GAA P10253 2/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
PLA2G2A P14555 1/20 0.34
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MCL1 Q07820 1/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
NPC1 O15118 1/20 0.33
TDP1 Q9NUW8 2/20 0.33
USP2 O75604 1/20 0.33
GABRP O00591 1/20 0.32
GABRD O14764 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL599521 0.79 DAO (0.33) KDM4EGAASMN1; SMN2
SCHEMBL11325534 0.73 RXFP1 (0.49) MAPTKDM4EALDH1A1GAAMEN1
SCHEMBL649606 0.72 AKR1C3 (0.41) ALDH1A1
SCHEMBL18029143 0.72 GPR17 (0.46) GPR17MAPTKDM4EALDH1A1GAA
SCHEMBL598456 0.71 KDM4E (0.59) GPR17FEN1MAPTKDM4EALDH1A1
SCHEMBL260657 0.71 CYP1A2 (0.40) MAPTSMN1; SMN2MEN1KMT2ATDP1
SCHEMBL11219094 0.68 PLA2G2A (0.35) MAPTALDH1A1GAAPLA2G2AMCL1
SCHEMBL2542691 0.68 GABRA1 (0.44) MAPTKDM4EALDH1A1GAASMN1; SMN2
SCHEMBL8298676 0.68 KDM4E (0.47) GPR17MAPTKDM4EALDH1A1GAA
SCHEMBL22609023 0.67 AHR (0.52) GPR17FEN1MAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8115014-B2 Ethynylindole compounds ONO Pharmaceuticals, Co., Ltd. (JP) 2012-02-14 US disclosed