SCHEMBL5983475

SCHEMBL5983475

CN(c1cccc(NC(=O)c2ccc(F)cc2F)n1)C1CCNCC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1F P30939 6/20 0.48
SMN1; SMN2 Q16637 2/20 0.41
TP53 P04637 2/20 0.41
NPC1 O15118 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
RAB9A P51151 1/20 0.41
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
CHRM5 P08912 1/20 0.39
DRD5 P21918 1/20 0.39
HTR1D P28221 1/20 0.39
HTR1E P28566 1/20 0.39
HTR7 P34969 1/20 0.39
OPRK1 P41145 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12020910 0.90 SLC6A2 (0.44) HTR1FNPC1RAB9AALDH1A1MEN1
SCHEMBL1197874 0.87 HTR1F (0.60) HTR1FALDH1A1LMNACHRM5DRD5
Hydrochloric Acid SCHEMBL5984136 0.87 HTR1F (0.51) HTR1FNPC1CYP1A2RAB9ACHRM5
SCHEMBL12021012 0.85 HTR1F (0.50) HTR1FNPC1RAB9AHTR1DHTR1E
Hydrochloric Acid SCHEMBL5983376 0.85 HTR1F (0.49) HTR1FNPC1RAB9AHTR1DHTR1E
SCHEMBL5983275 0.84 MEN1 (0.54) HTR1FNPC1CYP1A2RAB9ACHRM5
Hydrochloric Acid SCHEMBL5983739 0.80 CCNA2 (0.45) SMN1; SMN2TP53NPC1CYP1A2CYP2C19
Hydrochloric Acid SCHEMBL5983416 0.80 ALDH1A1 (0.53) SMN1; SMN2NPC1CYP1A2CYP2C19RAB9A
SCHEMBL5983353 0.79 FLT3 (0.43) HTR1FCHRM5DRD5HTR1DHTR1E
SCHEMBL5983472 0.79 MEN1 (0.43) HTR1FCHRM5DRD5HTR1DHTR1E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663971-A1 SUBSTITUTED 2-CARBONYLAMINO-6-PIPERIDINAMINOPYRIDINES AND SUBSTITUTED 1-CARBONYLAMINO-3-PIPERIDINAMINOBENZENES AS 5-HT1F AGONISTS Eli Lilly and Company (US) 2006-06-07 EP disclosed
WO-2005035499-A1 SUBSTITUTED 2-CARBONYLAMINO-6-PIPERIDINAMINOPYRIDINES AND SUBSTITUTED 1-CARBONYLAMINO-3-PIPERIDINAMINOBENZENES AS 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 2005-04-21 WO disclosed