SCHEMBL5990907

SCHEMBL5990907

CCc1ccc(O)c(-c2cccs2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.48
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44
TMIGD3 P0DMS9 2/20 0.41
ADORA2A P29274 2/20 0.41
ADORA1 P30542 2/20 0.41
MAPT P10636 6/20 0.41
KDM4E B2RXH2 1/20 0.41
TP53 P04637 1/20 0.41
THRB P10828 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
TDP1 Q9NUW8 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
LMNA P02545 2/20 0.40
RPS6KB2 Q9UBS0 1/20 0.40
ALDH1A1 P00352 5/20 0.40
GAA P10253 3/20 0.40
HSP90AA1 P07900 2/20 0.40
S1PR4 O95977 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5989750 0.88 TRPA1 (0.38) TRPA1CNR1CNR2TMIGD3ADORA2A
SCHEMBL23991290 0.81 BACE1 (0.58) CNR1CNR2TMIGD3ADORA2AADORA1
Hydrochloric Acid SCHEMBL23629396 0.80 BACE1 (0.56) CNR1CNR2MAPTKDM4ETP53
SCHEMBL29763176 0.78 TRPA1 (0.70) TRPA1CNR1CNR2MAPTKDM4E
SCHEMBL8047684 0.78 TRPA1 (0.70) TRPA1CNR1CNR2MAPTKDM4E
SCHEMBL14027112 0.78 RPS6KB2 (0.53) TMIGD3ADORA2AADORA1MAPTKDM4E
SCHEMBL5990688 0.78 ERN1 (0.47) MAPTKDM4ETP53SMN1; SMN2MEN1
SCHEMBL4124686 0.77 CSNK2A1 (0.42) ADORA2AADORA1MAPTKDM4ETP53
SCHEMBL27968468 0.74 MAPT (0.41) ADORA2AADORA1MAPTKDM4ETP53
SCHEMBL13996579 0.74 TRPA1 (0.46) TRPA1CNR1CNR2MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060257987-A1 Ppar modulators ELI LILLY AND COMPANY 2006-11-16 US disclosed
EP-1660428-A1 PPAR MODULATORS ELI LILLY AND COMPANY (US) 2006-05-31 EP disclosed
WO-2005019151-A1 PPAR MODULATORS ELI LILLY AND COMPANY (US) 2005-03-03 WO disclosed