SCHEMBL6001767

SCHEMBL6001767

COC(=O)CCCCC(C=O)Cc1ccccc1C#N

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.44
ALDH1A1 P00352 3/20 0.44
HPGD P15428 1/20 0.44
CNR2 P34972 2/20 0.39
PPARG P37231 2/20 0.38
GAA P10253 1/20 0.36
POLB P06746 1/20 0.36
PPARA Q07869 1/20 0.36
LMNA P02545 1/20 0.36
FFAR1 O14842 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
DPP4 P27487 1/20 0.35
FAP Q12884 1/20 0.35
DPP8 Q6V1X1 1/20 0.35
DPP9 Q86TI2 1/20 0.35
DPP7 Q9UHL4 1/20 0.35
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAOB P27338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6002358 0.82 TSHR (0.44) TSHRALDH1A1HPGDCNR2PPARG
SCHEMBL7094632 0.79 TSHR (0.52) TSHRALDH1A1HPGDCNR2GAA
SCHEMBL4837680 0.77 TSHR (0.53) TSHRALDH1A1HPGDCNR2GAA
SCHEMBL12255638 0.74 TSHR (0.56) TSHRALDH1A1HPGDCNR2GAA
SCHEMBL13443169 0.73 TSHR (0.54) TSHRALDH1A1PPARGPOLBLMNA
SCHEMBL3594770 0.71 CYP4A11 (0.43) TSHRALDH1A1HPGDGAALMNA
SCHEMBL1558841 0.71 ALDH1A1 (0.51) TSHRALDH1A1HPGDGAAPOLB
SCHEMBL28346434 0.70 ALDH1A1 (0.46) TSHRALDH1A1HPGDPPARGGAA
SCHEMBL9442266 0.69 TSHR (0.48) TSHRALDH1A1PPARGPOLBLMNA
SCHEMBL12851876 0.69 ALDH1A1 (0.47) TSHRALDH1A1HPGDGAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1655280-A1 Dicarboxylic acid derivates with pharmaceutical properties Bayer HealthCare AG (DE) 2006-05-10 EP disclosed
US-6864287-B1 Derivatives of dicarboxylic acid having pharmaceutical properties BAYER AKTIENGESELLSCHAFT (DE) 2005-03-08 US disclosed
EP-1216222-A2 NOVEL DERIVATIVES OF DICARBOXYLIC ACID HAVING PHARMACEUTICAL PROPERTIES Bayer Aktiengesellschaft (DE) 2002-06-26 EP disclosed
WO-2001019776-A2 NOVEL DERIVATIVES OF DICARBOXYLIC ACID HAVING PHARMACEUTICAL PROPERTIES BAYER AKTIENGESELLSCHAFT (DE) 2001-03-22 WO disclosed