SCHEMBL6002154

SCHEMBL6002154

COc1cc2c(cc1OC)C(N1CCN(C)CC1)CCC2

nearest known ligand 0.74

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 3/20 0.58
RAD52 P43351 1/20 0.57
DRD1 P21728 8/20 0.52
DRD2 P14416 4/20 0.52
HTR1A P08908 1/20 0.50
MAOA P21397 1/20 0.49
ABCB1 P08183 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31514974 0.85 CHRNA7 (0.76) CHRNA7RAD52DRD1DRD2HTR1A
SCHEMBL30932155 0.85 CHRNA7 (0.76) CHRNA7RAD52DRD1DRD2HTR1A
SCHEMBL30363169 0.85 CHRNA7 (0.76) CHRNA7RAD52DRD1DRD2HTR1A
SCHEMBL28765330 0.84 CHRNA7 (0.70) CHRNA7RAD52DRD1DRD2HTR1A
SCHEMBL30363191 0.84 CHRNA7 (0.70) CHRNA7RAD52DRD1DRD2HTR1A
SCHEMBL6406929 0.83 MTNR1B (0.49) CHRNA7DRD1DRD2
SCHEMBL21877880 0.82 RAD52 (0.61) CHRNA7RAD52DRD1DRD2HTR1A
SCHEMBL5320509 0.80 CHRNA7 (0.51) CHRNA7RAD52
SCHEMBL6001623 0.80 MTNR1B (0.70)
SCHEMBL6406088 0.79 MTNR1B (0.47) CHRNA7DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060166984-A1 Amino substituted benzo(hetero)cyclic derivatives BASF AKTIENGESELLSCHAFT (DE) 2006-07-27 US disclosed
EP-1603395-A2 AMINO SUBSTITUTED BENZO(HETERO)CYCLIC DERIVATIVES BASF AKTIENGESELLSCHAFT (DE) 2005-12-14 EP disclosed
WO-2004080170-A2 AMINO SUBSTITUTED BENZO(HETERO)CYCLIC DERIVATIVES BASF AKTIENGESELLSCHAFT (DE) 2004-09-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060166984-A1 Amino substituted benzo(hetero)cyclic derivatives CBR3, L3MBTL3, BRS3 CHRNA7 1146/4885RAD52 424/4885DRD1 1875/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.