SCHEMBL6002599

SCHEMBL6002599

C=CCC(CC)(C(N)=O)c1ccc(F)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.58
KCNN4 O15554 8/20 0.46
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45
KCNE1 P15382 1/20 0.36
KCNQ1 P51787 1/20 0.36
HTR7 P34969 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
KDM4E B2RXH2 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
RIPK1 Q13546 2/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
XBP1 P17861 1/20 0.33
MAPK1 P28482 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4005378 0.85 KCNN4 (0.57) HTTKCNN4ALDH1A1KCNE1KCNQ1
SCHEMBL4001444 0.77 ALDH1A1 (0.46) HTTKCNN4ALDH1A1TSHRHTR7
SCHEMBL2171612 0.72 KDM4E (0.44) HTTKCNN4ALDH1A1HTR7SMN1; SMN2
SCHEMBL9748549 0.71 ALDH1A1 (0.80) HTTALDH1A1TSHRSMN1; SMN2HDAC1
SCHEMBL8356496 0.70 KCNN4 (0.55) HTTKCNN4KCNE1KCNQ1SMN1; SMN2
SCHEMBL12833766 0.69 KCNN4 (0.38) HTTKCNN4ALDH1A1TSHRSMN1; SMN2
SCHEMBL3465944 0.69 HTT (0.81) HTTKCNN4ALDH1A1TSHRSMN1; SMN2
SCHEMBL3465945 0.69 HTT (0.81) HTTKCNN4ALDH1A1TSHRSMN1; SMN2
SCHEMBL1141842 0.68 OGG1 (0.42) HTTSMN1; SMN2HDAC3HDAC1HDAC2
SCHEMBL9721792 0.68 MAPT (0.46) HTTKCNN4ALDH1A1TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636221-A2 NEW AZETIDINE COMPOUNDS AstraZeneca AB (SE) 2006-03-22 EP disclosed
WO-2004110344-A2 NEW AZETIDINE COMPOUNDS ASTRAZENECA AB (SE) 2004-12-23 WO disclosed