SCHEMBL6002890

SCHEMBL6002890

Fc1ccc(-c2c[nH][c]n2)cc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.41
KMO O15229 2/20 0.38
ALDH1A1 P00352 2/20 0.37
CYP1A2 P05177 2/20 0.37
GAA P10253 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
MAOB P27338 1/20 0.36
TRPA1 O75762 2/20 0.36
TYMP P19971 1/20 0.35
CYP17A1 P05093 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
RAB9A P51151 3/20 0.35
KDM4E B2RXH2 2/20 0.35
MAPK1 P28482 1/20 0.35
IDO1 P14902 1/20 0.34
NPC1 O15118 2/20 0.34
TGFBR1 P36897 2/20 0.34
TOP1 P11387 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27776210 0.82 MPL (0.49) NOTUMKMOCYP11B1CYP11B2
SCHEMBL4046110 0.79 RAB9A (0.37) ALDH1A1RAB9AKDM4EMAPK1NPC1
SCHEMBL2093090 0.76 IDO1 (0.49) KMOALDH1A1MAOBRAB9AKDM4E
SCHEMBL4049874 0.75 NOTUM (0.34) NOTUM
SCHEMBL1202001 0.75 NOTUM (0.42) NOTUMALDH1A1CYP1A2GAARAB9A
SCHEMBL27584582 0.75 METAP2 (0.42) ALDH1A1GAARAB9AKDM4EMAPK1
SCHEMBL17626110 0.74 AHR (0.46) NOTUMKMOALDH1A1GAARAB9A
SCHEMBL1319204 0.73 IDO1 (0.49) NOTUMKMOALDH1A1GAAKDM4E
SCHEMBL4044388 0.73 TGFBR1 (0.33) ALDH1A1RAB9AKDM4EIDO1TGFBR1
SCHEMBL4050038 0.73 CYP1A2 (0.47) ALDH1A1CYP1A2CYP2C9CYP2C19MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678185-A1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-07-12 EP disclosed
WO-2005042542-A1 2,3-DIHYDRO-6-NITROIMIDAZO (2,1-B) OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2005-05-12 WO disclosed