SCHEMBL6002962

SCHEMBL6002962

CCc1csc2c(Cl)cccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.38
CYP2A6 P11509 3/20 0.38
DRD3 P35462 2/20 0.37
LMNA P02545 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
PGR P06401 1/20 0.37
CHRM2 P08172 1/20 0.37
HTR1A P08908 1/20 0.37
ADRA2A P08913 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
AR P10275 1/20 0.37
CHRM1 P11229 1/20 0.37
IDO1 P14902 1/20 0.37
DRD1 P21728 1/20 0.37
TBXA2R P21731 1/20 0.37
ACHE P22303 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4664840 0.83 CYP2A6 (0.39) CYP1A2CYP2A6DRD3LMNACYP3A4
SCHEMBL2090742 0.81 CYP2A6 (0.38) CYP1A2CYP2A6DRD3LMNACYP3A4
SCHEMBL3985620 0.81 CYP2A6 (0.38) CYP1A2CYP2A6DRD3LMNACYP3A4
SCHEMBL8587770 0.79 TAAR1 (0.50) CYP1A2CYP2A6DRD3LMNACYP3A4
SCHEMBL17038612 0.78 F2RL1 (0.36) CYP2A6LMNASLC6A4MIFGABRA1
SCHEMBL6299526 0.78 GABRA1 (0.42) CYP1A2CYP2A6CYP2D6CYP2C19GABRA1
SCHEMBL29908309 0.75 CYP2A6 (0.42) CYP1A2CYP2A6MIFMCL1GAA
SCHEMBL787846 0.75 CYP2A6 (0.42) CYP1A2CYP2A6MIFMCL1GAA
SCHEMBL6305533 0.74 CLCN2 (0.43) LMNACYP2C9TDP1MEN1RAB9A
SCHEMBL2091808 0.74 CYP1A2 (0.34) CYP1A2CYP2A6DRD3LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7323433-B2 R-(-)-1-[2-(7-chlorobenzo[b]thiopen-3-yl-methoxy)-2-(2,4-dichlorophenyl)-ethyl]-1H-imidazole FERRER INTERNACIONAL, S.A. (ES) 2008-01-29 US disclosed
EP-1678185-A1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-07-12 EP disclosed
WO-2005042542-A1 2,3-DIHYDRO-6-NITROIMIDAZO (2,1-B) OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2005-05-12 WO disclosed